143113-45-5
Chemical Structure
BQ-3020
- CAS 番号: 143113-45-5
- Formula:C96H140N20O24S
- Molecular Weight:1990.32
InChIKey: CUZUEERSGQQGSO-LQTSPBQXSA-N
SMILES: O=C(C)N[C@@H](CC(C)C)C(N[C@H](CCSC)C(N[C@@H](CC(O)=O)C(N[C@H](CCCCN)C(N[C@@H](CCC(O)=O)C(N[C@H](C)C(N[C@@H](C(C)C)C(N[C@H](CC1=CC=C(O)C=C1)C(N[C@H](C(N[C@H](C)C(N[C@@H](CC2=CN=CN2)C(N[C@H](CC(C)C)C(N[C@@H](CC(O)=O)C(N[C@]([C@@H](C)CC)([H])C(N[C@@]([C@@H](C)CC)(C(N[C@H](CC3=CNC4=C3C=CC=C4)C=O)=O)[H])=O)=O)=O)=O)=O)=O)CC5=CC=CC=C5)=O)=O)=O)=O)=O)=O)=O)=O
Biological Activity: BQ-3020 is a selective endothelin receptor (ETB receptor) agonist that displaces [125I] ET-1 binding to ETB receptors, with an IC50 value of 0.2 nM. BQ-3020 elicits vasoconstriction in the rabbit pulmonary artery. BQ-3020 makes relaxation of the pig urinary bladder neck and can be used for cardiovascular disease research12.
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BQ-3020 | BQ-3020 is a selective endothelin receptor (ETB receptor) agonist that displaces [125I] ET-1 binding to ETB receptors, with an IC50 value of 0.2 nM. BQ-3020 elicits vasoconstriction in the rabbit pulmonary artery. BQ-3020 makes relaxation of the pig urinary bladder neck and can be used for cardiovascular disease research12. | |||||||||||||||||||||
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