150586-58-6
150586-58-6
Chemical Structure
Fipamezole
Synonym(s): MPV 1730; JP-1730
- CAS No.: 150586-58-6
- Formula:C14H15FN2
- Molecular Weight:230.28
IUPAC Name: 5-(2-ethyl-5-fluoro-2,3-dihydro-1H-inden-2-yl)-1H-imidazole
InChIKey: KXSUAWAUCNFBQJ-UHFFFAOYSA-N
SMILES: FC1=CC=C2C(CC(C2)(CC)C3=CN=CN3)=C1
Biological Activity: Fipamezole (MPV 1730; JP-1730) is a potent and orally active α2-adrenergic receptor antagonist with Ki values of 9.2 nM, 17 nM, and 55 nM for human α2A, α2B, and α2C, receptors, respectively. Fipamezole is an anti-dyskinetic agent, and can be used for the study of Parkinson's disease[1].
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Fipamezole | Fipamezole (MPV 1730; JP-1730) is a potent and orally active α2-adrenergic receptor antagonist with Ki values of 9.2 nM, 17 nM, and 55 nM for human α2A, α2B, and α2C, receptors, respectively. Fipamezole is an anti-dyskinetic agent, and can be used for the study of Parkinson's disease. | |||||||||||||||||||||
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References
Keywords
