152241-24-2
152241-24-2
Chemical Structure
GT-2016
- CAS No.: 152241-24-2
- Formula:C19H31N3O
- Molecular Weight:317.47
IUPAC Name: 1-(4-(1H-imidazol-4-yl)piperidin-1-yl)-5-cyclohexylpentan-1-one
InChIKey: YTCGNPGLMAECND-UHFFFAOYSA-N
SMILES: O=C(N1CCC(C2=CNC=N2)CC1)CCCCC3CCCCC3
Biological Activity: GT-2016 is a potent, selective, and brain penetrant histamine H3 receptor antagonist with a Ki of 43.8 nM. GT-2016 displays selectivity against H1 and H2 receptors, and has non-active against histamine methyltransferase[1].
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GT-2016 | GT-2016 is a potent, selective, and brain penetrant histamine H3 receptor antagonist with a Ki of 43.8 nM. GT-2016 displays selectivity against H1 and H2 receptors, and has non-active against histamine methyltransferase. | |||||||||||||||||||||
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References
Keywords
