1572922-53-2
Chemical Structure
5-Hydroxy saxagliptin-13C,d2-2 hydrochloride
- CAS No.: 1572922-53-2
- Formula:C1713CH24D2ClN3O3
- Molecular Weight:370.88
InChIKey: WCCKQMJRTRWMMX-HHZNFPBZSA-N
SMILES: O=C(N1[C@]2([H])[C@@](C[C@H]1C#N)([H])[13C]2([2H])[2H])[C@H](C34CC5(CC(C3)(CC(C5)C4)O)O)N.Cl
Biological Activity: 5-Hydroxy saxagliptin-13C,d2-2 hydrochloride is the 13C- and deuterium labeled 5-Hydroxy saxagliptin hydrochloride. 5-Hydroxy saxagliptin hydrochloride is an active metabolite of Saxagliptin (HY-10285) and a potent and selective DPP-4 inhibitor. 5-Hydroxy saxagliptin hydrochloride has Ki values of 2.6 nM and 2.9 nM for humans and cynomolgus monkeys, respectively. 5-Hydroxy saxagliptin hydrochloride can be used in the research of type 2 diabetes mellitus[1].
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5-Hydroxy saxagliptin-13C,d2-2 hydrochloride | 5-Hydroxy saxagliptin-13C,d2-2 hydrochloride is the 13C- and deuterium labeled 5-Hydroxy saxagliptin hydrochloride. 5-Hydroxy saxagliptin hydrochloride is an active metabolite of Saxagliptin (HY-10285) and a potent and selective DPP-4 inhibitor. 5-Hydroxy saxagliptin hydrochloride has Ki values of 2.6 nM and 2.9 nM for humans and cynomolgus monkeys, respectively. 5-Hydroxy saxagliptin hydrochloride can be used in the research of type 2 diabetes mellitus. | |||||||||||||||||||||
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