185954-27-2
185954-27-2
Chemical Structure
Tofimilast
- CAS No.: 185954-27-2
- Formula:C18H21N5S
- Molecular Weight:339.46
IUPAC Name: 9-cyclopentyl-7-ethyl-3-(thiophen-2-yl)-6,9-dihydro-5H-pyrazolo[3,4-c][1,2,4]triazolo[4,3-a]pyridine
InChIKey: DHCOPPHTVOXDKU-UHFFFAOYSA-N
SMILES: CCC1=NN(C2=C1CCN3C2=NN=C3C4=CC=CS4)C5CCCC5
Biological Activity: Tofimilast is an inhibitor of Phosphodiesterase 4 (PDE4) with an IC50 of 0.14 μM. Tofimilast exerts its anti-inflammatory effects by inhibiting the activity of PDE4, thereby increasing intracellular levels of cAMP[1].
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Tofimilast | Tofimilast is an inhibitor of Phosphodiesterase 4 (PDE4) with an IC50 of 0.14 μM. Tofimilast exerts its anti-inflammatory effects by inhibiting the activity of PDE4, thereby increasing intracellular levels of cAMP. | |||||||||||||||||||||
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References
Keywords
