2040401-92-9
Chemical Structure
BI-6901
- CAS No.: 2040401-92-9
- Formula:C23H27N5O3S
- Molecular Weight:453.56
IUPAC Name: (R)-N-(4-(2-cyano-1H-pyrrol-1-yl)-1-(4-methylpiperidin-1-yl)-1-oxobutan-2-yl)-1H-indole-4-sulfonamide
InChIKey: BRJXJOWXAFLRTE-OAQYLSRUSA-N
SMILES: O=S(C1=CC=CC2=C1C=CN2)(N[C@@H](C(N3CCC(C)CC3)=O)CCN4C(C#N)=CC=C4)=O
Biological Activity: BI 6901 is a potent, selective CCR10 antagonist (pIC50=9.0). BI 6901 shows high selectivity over other GPCRs, including a number of other chemokine receptors. BI 6901 is efficacious in the murine DNFB model of contact hypersensitivity and can be used for inflammation research[1].
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BI-6901 | 99.76% | BI 6901 is a potent, selective CCR10 antagonist (pIC50=9.0). BI 6901 shows high selectivity over other GPCRs, including a number of other chemokine receptors. BI 6901 is efficacious in the murine DNFB model of contact hypersensitivity and can be used for inflammation research. | ||||||||||||||||||||
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Keywords
