208993-54-8
208993-54-8
Chemical Structure
Fiduxosin
- CAS No.: 208993-54-8
- Formula:C30H29N5O4S
- Molecular Weight:555.65
IUPAC Name: 3-(4-((3aR,9bR)-9-methoxy-1,3a,4,9b-tetrahydrochromeno[3,4-c]pyrrol-2(3H)-yl)butyl)-8-phenylpyrazino[2',3':4,5]thieno[3,2-d]pyrimidine-2,4(1H,3H)-dione
InChIKey: WDTAYDBPNYFWDR-WOJBJXKFSA-N
SMILES: O=C(N1CCCCN2C[C@]3([H])[C@](COC4=CC=CC(OC)=C34)([H])C2)C5=C(NC1=O)C6=NC(C7=CC=CC=C7)=CN=C6S5
Biological Activity: Fiduxosin is a potent α1-adrenoceptor antagonist, with Ki of 0.160 nM, 24.9 nM, and 0.920 nM for α1a-, α1b-, and α1d-adrenoceptors, respectively.
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Fiduxosin | Fiduxosin is a potent α1-adrenoceptor antagonist, with Ki of 0.160 nM, 24.9 nM, and 0.920 nM for α1a-, α1b-, and α1d-adrenoceptors, respectively. | |||||||||||||||||||||
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