2138814-32-9
2138814-32-9
Chemical Structure
GSK3004774
- CAS No.: 2138814-32-9
- Formula:C32H40N4O3
- Molecular Weight:528.69
IUPAC Name: 1-(3-(4-((S)-3-(((R)-1-(naphthalen-1-yl)ethyl)amino)pyrrolidin-1-yl)benzamido)propyl)piperidine-4-carboxylic acid
InChIKey: HBTVUVNVTSSIHP-KCWPFWIISA-N
SMILES: O=C(NCCCN1CCC(C(O)=O)CC1)C(C=C2)=CC=C2N(CC3)C[C@H]3N[C@H](C)C4=CC=CC5=C4C=CC=C5
Biological Activity: GSK3004774 is a potent, nonabsorbable agonist of CaSR, with an pEC50 of 7.3, 6.6 and 6.5 for human, mouse and rat CaSR, respectively. GSK3004774 shows an EC50 of 50 nM for human CaSR[1].
| Cat. No. | Product Name | Purity | Description | Pricing | |||||||||||||||||||
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GSK3004774 | 99.09% | GSK3004774 is a potent, nonabsorbable agonist of CaSR, with an pEC50 of 7.3, 6.6 and 6.5 for human, mouse and rat CaSR, respectively. GSK3004774 shows an EC50 of 50 nM for human CaSR. | ||||||||||||||||||||
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GSK3004774 (Standard) | GSK3004774 (Standard) is the analytical standard of GSK3004774 (HY-107773). This product is intended for research and analytical applications. GSK3004774 is a potent, nonabsorbable agonist of CaSR, with an pEC50 of 7.3, 6.6 and 6.5 for human, mouse and rat CaSR, respectively. GSK3004774 shows an EC50 of 50 nM for human CaSR. | |||||||||||||||||||||
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References
Keywords
