1. GPCR/G Protein
  2. CaSR

GSK3004774 

Cat. No.: HY-107773
Handling Instructions

GSK3004774 is a potent, nonabsorbable agonist of CaSR, with an pEC50 of 7.3, 6.6 and 6.5 for human, mouse and rat CaSR, respectively. GSK3004774 shows an EC50 of 50 nM for human CaSR.

For research use only. We do not sell to patients.

GSK3004774 Chemical Structure

GSK3004774 Chemical Structure

CAS No. : 2138814-32-9

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Description

GSK3004774 is a potent, nonabsorbable agonist of CaSR, with an pEC50 of 7.3, 6.6 and 6.5 for human, mouse and rat CaSR, respectively. GSK3004774 shows an EC50 of 50 nM for human CaSR[1].

References
Molecular Weight

528.69

Formula

C₃₂H₄₀N₄O₃

CAS No.

2138814-32-9

SMILES

O=C(NCCCN1CCC(C(O)=O)CC1)C(C=C2)=CC=C2N(CC3)C[[email protected]]3N[[email protected]](C)C4=CC=CC5=C4C=CC=C5

Storage

Please store the product under the recommended conditions in the Certificate of Analysis.

Shipping

Room temperature in continental US; may vary elsewhere

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This equation is commonly abbreviated as: C1V1 = C2V2

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C1   V1   C2   V2

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Product Name:
GSK3004774
Cat. No.:
HY-107773
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GSK3004774

Cat. No.: HY-107773