2159137-02-5
2159137-02-5
Chemical Structure
GSK097
- CAS No.: 2159137-02-5
- Formula:C19H21N3O3
- Molecular Weight:339.39
IUPAC Name: 6-((S)-hydroxy(phenyl)methyl)-N2-methyl-N4-((1S,2S)-2-methylcyclopropyl)pyridine-2,4-dicarboxamide
InChIKey: OJSKWCXPUVTNCF-YLVFBTJISA-N
SMILES: O=C(C1=NC([C@@H](O)C2=CC=CC=C2)=CC(C(N[C@@H]3[C@@H](C)C3)=O)=C1)NC
Biological Activity: GSK097 is a potent and selective Inhibitor of the second bromodomain (BD2) of the bromodomain and extra-terminal domain (BET) proteins. GSK097 displays 2000-fold selective for BD2 over BD1 (BRD4 data) with >1 mg/mL solubility in FaSSIF media[1].
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GSK097 | GSK097 is a potent and selective Inhibitor of the second bromodomain (BD2) of the bromodomain and extra-terminal domain (BET) proteins. GSK097 displays 2000-fold selective for BD2 over BD1 (BRD4 data) with >1 mg/mL solubility in FaSSIF media. | |||||||||||||||||||||
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References
Keywords
