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  3. GSK097

GSK097 

Cat. No.: HY-132232
Handling Instructions

GSK097 is a potent and selective Inhibitor of the second bromodomain (BD2) of the bromodomain and extra-terminal domain (BET) proteins. GSK097 displays 2000-fold selective for BD2 over BD1 (BRD4 data) with >1 mg/mL solubility in FaSSIF media.

For research use only. We do not sell to patients.

GSK097 Chemical Structure

GSK097 Chemical Structure

CAS No. : 2159137-02-5

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Description

GSK097 is a potent and selective Inhibitor of the second bromodomain (BD2) of the bromodomain and extra-terminal domain (BET) proteins. GSK097 displays 2000-fold selective for BD2 over BD1 (BRD4 data) with >1 mg/mL solubility in FaSSIF media[1].

In Vitro

GSK097 displays pIC50s 7.4, 8.0, 7.6, and 7.9 for BRD2 BD2, BRD3 BD2, BRD4 BD2 and BRDT BD2, respectively[1].

MCE has not independently confirmed the accuracy of these methods. They are for reference only.

Molecular Weight

339.39

Formula

C₁₉H₂₁N₃O₃

CAS No.
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Storage

Please store the product under the recommended conditions in the Certificate of Analysis.

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GSK097
Cat. No.:
HY-132232
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