2250025-98-8
Chemical Structure
BRK inhibitor P21d hydrochloride
- CAS No.: 2250025-98-8
- Formula:C23H23ClFN7O2
- Molecular Weight:483.93
IUPAC Name: (4-((6-cyclopropyl-3-(1H-pyrazol-4-yl)imidazo[1,2-a]pyrazin-8-yl)amino)-3-fluorophenyl)(morpholino)methanone hydrochloride
InChIKey: GWHGHKMCIUENCZ-UHFFFAOYSA-N
SMILES: O=C(C1=CC=C(NC2=NC(C3CC3)=CN4C2=NC=C4C5=CNN=C5)C(F)=C1)N6CCOCC6.[H]Cl
Biological Activity: BRK inhibitor P21d hydrochloride is a potent breast tumor kinase (BRK/PTK6) inhibitor with an IC50 of 30 nM. BRK inhibitor P21d hydrochloride inhibits p-SAM68 with an IC50 of 52 nM. BRK inhibitor P21d hydrochloride can be used to evaluate the in vivo activity of BRK inhibitors in xenograft breast tumor models[1].
| Cat. No. | Product Name | Purity | Description | Pricing | |||||||||||||||||||
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BRK inhibitor P21d hydrochloride | 99.77% | BRK inhibitor P21d hydrochloride is a potent breast tumor kinase (BRK/PTK6) inhibitor with an IC50 of 30 nM. BRK inhibitor P21d hydrochloride inhibits p-SAM68 with an IC50 of 52 nM. BRK inhibitor P21d hydrochloride can be used to evaluate the in vivo activity of BRK inhibitors in xenograft breast tumor models. | ||||||||||||||||||||
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Keywords
