225120-65-0
225120-65-0
Chemical Structure
Cathepsin inhibitor 1
- CAS No.: 225120-65-0
- Formula:C20H24ClN5O2
- Molecular Weight:401.89
IUPAC Name: (S)-3-(tert-butyl)-N-(3-(3-chlorophenyl)-1-((cyanomethyl)amino)-1-oxopropan-2-yl)-1-methyl-1H-pyrazole-5-carboxamide
InChIKey: MZRVIHRERYCHBL-HNNXBMFYSA-N
SMILES: O=C(C1=CC(C(C)(C)C)=NN1C)N[C@@H](CC2=CC=CC(Cl)=C2)C(NCC#N)=O
Biological Activity: Cathepsin inhibitor 1 (Compound 25) is a potent and selective inhibitor of Cathepsin, with pIC50s of 7.9, 6.7, 6.0, 5.5 and 5.2 for CatL, CatL2, CatS, CatK, and CatB, respectively. Cathepsin inhibitor 1 is promising for research of osteoarthritis[1].
| Cat. No. | Nom du produit | Pureté | Description | Pricing | |||||||||||||||||||
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Cathepsin inhibitor 1 | 99.28% | Cathepsin inhibitor 1 (Compound 25) is a potent and selective inhibitor of Cathepsin, with pIC50s of 7.9, 6.7, 6.0, 5.5 and 5.2 for CatL, CatL2, CatS, CatK, and CatB, respectively. Cathepsin inhibitor 1 is promising for research of osteoarthritis. | ||||||||||||||||||||
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