2259640-87-2
2259640-87-2
Chemical Structure
CBP/p300-IN-17
- CAS No.: 2259640-87-2
- Formula:C25H28N4O3
- Molecular Weight:432.51
IUPAC Name: (R)-N-(1H-indazol-4-yl)-1-(1-(4-methoxyphenyl)cyclopentane-1-carbonyl)pyrrolidine-2-carboxamide
InChIKey: KRGAGJKQQRBFEC-JOCHJYFZSA-N
SMILES: O=C([C@@H]1N(C(C2(C3=CC=C(OC)C=C3)CCCC2)=O)CCC1)NC4=CC=CC5=C4C=NN5
Biological Activity: CBP/p300-IN-17 (compound 7) is a potent EP300/CBP HAT inhibitor with IC50s of 0.18, 0.69 µM for HAT EP300 and LK2 H3K27, respectively[1].
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CBP/p300-IN-17 | CBP/p300-IN-17 (compound 7) is a potent EP300/CBP HAT inhibitor with IC50s of 0.18, 0.69 µM for HAT EP300 and LK2 H3K27, respectively. | |||||||||||||||||||||
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