1. Epigenetics
  2. Histone Acetyltransferase
  3. CBP/p300-IN-17

CBP/p300-IN-17 

Cat. No.: HY-143441
Handling Instructions

CBP/p300-IN-17 (compound 7) is a potent EP300/CBP HAT inhibitor with IC50s of 0.18, 0.69 µM for HAT EP300 and LK2 H3K27, respectively.

For research use only. We do not sell to patients.

CBP/p300-IN-17 Chemical Structure

CBP/p300-IN-17 Chemical Structure

CAS No. : 2259640-87-2

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Description

CBP/p300-IN-17 (compound 7) is a potent EP300/CBP HAT inhibitor with IC50s of 0.18, 0.69 µM for HAT EP300 and LK2 H3K27, respectively[1].

IC50 & Target[1]

EP300

0.18 μM (IC50)

LK2 H3K27

0.69 μM (IC50)

Molecular Weight

432.51

Formula

C25H28N4O3

CAS No.
SMILES

O=C([[email protected]@H]1N(C(C2(C3=CC=C(OC)C=C3)CCCC2)=O)CCC1)NC4=CC=CC5=C4C=NN5

Shipping

Room temperature in continental US; may vary elsewhere.

Storage

Please store the product under the recommended conditions in the Certificate of Analysis.

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Product Name:
CBP/p300-IN-17
Cat. No.:
HY-143441
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