CBP/p300-IN-17
CBP/p300-IN-17 (compound 7) is a potent EP300/CBP HAT inhibitor with IC50s of 0.18, 0.69 µM for HAT EP300 and LK2 H3K27, respectively.
For research use only. We do not sell to patients.
- CAS No.: 2259640-87-2
- Formula: C25H28N4O3
- Molecular Weight:432.51
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Storage:
Please store the product under the recommended conditions in the Certificate of Analysis.
Biological Activity
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EP300 .18 μM (IC50) |
LK2 H3K27 0.69 μM (IC50) |
Chemical Information
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CAS No. 2259640-87-2
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Molecular Weight 432.51
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Formula C25H28N4O3
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SMILES
O=C([C@@H]1N(C(C2(C3=CC=C(OC)C=C3)CCCC2)=O)CCC1)NC4=CC=CC5=C4C=NN5
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Shipping
Room temperature in continental US; may vary elsewhere.
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Storage
Please store the product under the recommended conditions in the Certificate of Analysis.
Purity & Documentation
References
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)