2332897-85-3
Chemical Structure
Nav1.1 activator 1
- CAS No.: 2332897-85-3
- Formula:C24H23F3N4O
- Molecular Weight:440.46
IUPAC Name: (S)-4-(2,5-difluorophenyl)-2-(3-fluoropyrrolidin-1-yl)-N-(6-isopropylpyridin-3-yl)nicotinamide
InChIKey: HRGJTEFGFUJXIF-INIZCTEOSA-N
SMILES: O=C(C1=C(C2=CC(F)=CC=C2F)C=CN=C1N3C[C@@H](F)CC3)NC4=CC=C(C(C)C)N=C4
Biological Activity: Nav1.1 activator 1 (compound 4), a highly potent Nav1.1 activator with BBB penetration, increases decay time constant (tau) of Nav1.1 currents at 0.03 μM along with significant selectivity against Nav1.2, Nav1.5, and Nav1.6[1].
| Cat. No. | Product Name | Purity | Description | Pricing | |||||||||||||||||||
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Nav1.1 activator 1 | 98.98% | Nav1.1 activator 1 (compound 4), a highly potent Nav1.1 activator with BBB penetration, increases decay time constant (tau) of Nav1.1 currents at 0.03 μM along with significant selectivity against Nav1.2, Nav1.5, and Nav1.6. | ||||||||||||||||||||
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