2556833-57-7
2556833-57-7
Chemical Structure
mGAT3/4-IN-1
- CAS No.: 2556833-57-7
- Formula:C26H31ClN2O2S2
- Molecular Weight:503.12
IUPAC Name: 2-((4,4-bis(3-methylthiophen-2-yl)but-3-en-1-yl)(methyl)amino)-N-(2-chlorobenzyl)-4-hydroxybutanamide
InChIKey: IJIMBHRRVMFBCK-UHFFFAOYSA-N
SMILES: O=C(C(CCO)N(CC/C=C(C1=C(C)C=CS1)\C2=C(C)C=CS2)C)NCC3=C(Cl)C=CC=C3
Biological Activity: mGAT3/4-IN-1 (compound 19b) is a potent mGAT3/mGAT4 inhibitor, with pIC50 values of 5.31 and 5.24, respectively. mGAT3/4-IN-1 exhibits a significant tactile allodynia reduction in diabetic neuropathic mice[1].
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mGAT3/4-IN-1 | mGAT3/4-IN-1 (compound 19b) is a potent mGAT3/mGAT4 inhibitor, with pIC50 values of 5.31 and 5.24, respectively. mGAT3/4-IN-1 exhibits a significant tactile allodynia reduction in diabetic neuropathic mice. | |||||||||||||||||||||
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References
Keywords
