2641601-66-1

PROTAC EZH2 Degrader-26 Chemical Structure
2641601-66-1

Chemical Structure

PROTAC EZH2 Degrader-26

  • CAS No.: 2641601-66-1
  • Formula:C52H63N7O8
  • Molecular Weight:914.10

InChIKey: LRSUGMPLWWDHBW-UHFFFAOYSA-N

SMILES: CC1=C(C=C(C=C1N(CC)C2CCOCC2)C3=CC=C(C=C3)CN4CCN(CC4)CCCCCOC5=C(C6=CC=C5)C(N(C6=O)C7CCC(NC7=O)=O)=O)C(NCC8=C(C=C(NC8=O)C)C)=O

Biological Activity: PROTAC EZH2 Degrader-26 (compound 11) is an EZH2 degrader developed based on PROTAC technology. PROTAC EZH2 Degrader-26 has an IC50 of 5.80 nM against EZH2. PROTAC EZH2 Degrader-26 exhibits micromolar-level enzyme inhibitory activity against EZH1, with an EZH1 IC50 of 0.06 μM[1].

Cat. No. Product Name Purity Description Pricing
HY-181327 		PROTAC EZH2 Degrader-26 PROTAC EZH2 Degrader-26 (compound 11) is an EZH2 degrader developed based on PROTAC technology. PROTAC EZH2 Degrader-26 has an IC50 of 5.80 nM against EZH2. PROTAC EZH2 Degrader-26 exhibits micromolar-level enzyme inhibitory activity against EZH1, with an EZH1 IC50 of 0.06 μM.
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