2761146-51-2
2761146-51-2
Chemical Structure
VPC-13789
- CAS No.: 2761146-51-2
- Formula:C21H16F3N3O
- Molecular Weight:383.37
IUPAC Name: N-isopropyl-2-(5,6,7-trifluoro-1H-indol-3-yl)quinoline-5-carboxamide
InChIKey: FMNAWYZSFUYYRV-UHFFFAOYSA-N
SMILES: O=C(C1=C2C=CC(C3=CNC4=C3C=C(F)C(F)=C4F)=NC2=CC=C1)NC(C)C
Biological Activity: VPC-13789 is a potent, selective, and orally bioavailable antiandrogen. VPC-13789 can be used for the research of castration-resistant prostate cancer (CRPC) therapeutics. VPC-13789 inhibits androgen receptor (AR) transcriptional activity in LNCaP cells (IC50=0.19 μM)[1].
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VPC-13789 | VPC-13789 is a potent, selective, and orally bioavailable antiandrogen. VPC-13789 can be used for the research of castration-resistant prostate cancer (CRPC) therapeutics. VPC-13789 inhibits androgen receptor (AR) transcriptional activity in LNCaP cells (IC50=0.19 μM). | |||||||||||||||||||||
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