2. Vitamin D Related/Nuclear Receptor
  3. Androgen Receptor
  4. VPC-13789

VPC-13789 is a potent, selective, and orally bioavailable antiandrogen. VPC-13789 can be used for the research of castration-resistant prostate cancer (CRPC) therapeutics. VPC-13789 inhibits androgen receptor (AR) transcriptional activity in LNCaP cells (IC50=0.19 μM).

For research use only. We do not sell to patients.

VPC-13789 Chemical Structure

VPC-13789 Chemical Structure

CAS No. : 2761146-51-2

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VPC-13789 Related Antibodies

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Description

VPC-13789 is a potent, selective, and orally bioavailable antiandrogen. VPC-13789 can be used for the research of castration-resistant prostate cancer (CRPC) therapeutics. VPC-13789 inhibits androgen receptor (AR) transcriptional activity in LNCaP cells (IC50=0.19 μM)[1].

Molecular Weight

383.37

Formula

C21H16F3N3O
CAS No.
SMILES

O=C(C1=C2C=CC(C3=CNC4=C3C=C(F)C(F)=C4F)=NC2=CC=C1)NC(C)C
Shipping

Room temperature in continental US; may vary elsewhere.
Storage

Please store the product under the recommended conditions in the Certificate of Analysis.
Purity & Documentation
References
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VPC-13789 Related Classifications

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Help & FAQs
  • Do most proteins show cross-species activity?

    Species cross-reactivity must be investigated individually for each product. Many human cytokines will produce a nice response in mouse cell lines, and many mouse proteins will show activity on human cells. Other proteins may have a lower specific activity when used in the opposite species.

Keywords:

VPC-137892761146-51-2VPC13789VPC 13789Androgen Receptororally bioavailable;antiandrogen;castration-resistant prostate cancer;CRPC;androgen receptorInhibitorinhibitorinhibit

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HY-139970
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