2841457-05-2
2841457-05-2
Chemical Structure
5-HT2CR agonist 2
- CAS No.: 2841457-05-2
- Formula:C17H17Cl2NO2
- Molecular Weight:338.23
InChIKey: HDPQZPNMAUPPFG-UHFFFAOYSA-N
SMILES: COC1=C(C=C2C3=C1C4=C(CC3NCC2)C=CC=C4Cl)O.Cl
Biological Activity: 5-HT2CR agonist 2 (Compound 16k) is a selective, blood-brain barrier-penetrating and Gq-biased 5-HT2CR agonist, with an EC50 of 36 nM. 5-HT2CR agonist 2 attenuates MK801 (HY-15084B)-induced hyperlocomotion and reverses Phencyclidine-induced hyperlocomotor activity[1].
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5-HT2CR agonist 2 | 5-HT2CR agonist 2 (Compound 16k) is a selective, blood-brain barrier-penetrating and Gq-biased 5-HT2CR agonist, with an EC50 of 36 nM. 5-HT2CR agonist 2 attenuates MK801 (HY-15084B)-induced hyperlocomotion and reverses Phencyclidine-induced hyperlocomotor activity. | |||||||||||||||||||||
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