3033296-80-6
Chemical Structure
CYP121A1-IN-1
- CAS No.: 3033296-80-6
- Formula:C22H20N4O
- Molecular Weight:356.42
IUPAC Name: 1-(3,4-dichlorophenyl)-8-methyl-N-(2-(methylamino)ethyl)-9H-pyrido[3,4-b]indole-3-carboxamide hydrochloride
InChIKey: IDUIVCFNXSKLPB-UHFFFAOYSA-N
SMILES: C12=CC=CC=C1N(C3=NC=CC(CCC4=CNC5=C4C=CC=C5)=N3)CCO2
Biological Activity: CYP121A1-IN-1 is a potent CYP121A1 inhibitor with favorable activity against Mycobacterium tuberculosis (H37Rv MIC90～6.25 μM, ～2.2 μg/mL). CYP121A1-IN-1 can markedly reduce the production of mycocyclosin via inhibiting the CYP121A1 mediated turnover of cyclo(l-tyrosyl-l-tyrosyl) to mycocyclosin[1].
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CYP121A1-IN-1 | CYP121A1-IN-1 is a potent CYP121A1 inhibitor with favorable activity against Mycobacterium tuberculosis (H37Rv MIC90～6.25 μM, ～2.2 μg/mL). CYP121A1-IN-1 can markedly reduce the production of mycocyclosin via inhibiting the CYP121A1 mediated turnover of cyclo(l-tyrosyl-l-tyrosyl) to mycocyclosin. | |||||||||||||||||||||
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Keywords
