CYP121A1-IN-1
CYP121A1-IN-1 is a potent CYP121A1 inhibitor with favorable activity against Mycobacterium tuberculosis (H37Rv MIC90～6.25 μM, ～2.2 μg/mL). CYP121A1-IN-1 can markedly reduce the production of mycocyclosin via inhibiting the CYP121A1 mediated turnover of cyclo(l-tyrosyl-l-tyrosyl) to mycocyclosin.
For research use only. We do not sell to patients.
- CAS No.: 3033296-80-6
- Formula: C22H20N4O
- Molecular Weight:356.42
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Storage:
Please store the product under the recommended conditions in the Certificate of Analysis.
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Biological Activity
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Chemical Information
- Purity & Documentation
- References
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Help & FAQs
Biological Activity
MIC90: 6.25 μM, 2.2 μg/mL (H37Rv)[1]
CYP121A1-IN-1 (compound 61) (0.78-400 μM; one week for c7H9 and 7H9-Low BSA media or two weeks for MMM-Ch medium) has favorable activity against Mtb strain H37Rv (MIC90～6.25 μM, ～2.2 μg/mL)[1].
MedChemExpress (MCE) has not independently confirmed the accuracy of these methods. They are for reference only.
Chemical Information
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CAS No. 3033296-80-6
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Molecular Weight 356.42
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Formula C22H20N4O
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SMILES
C12=CC=CC=C1N(C3=NC=CC(CCC4=CNC5=C4C=CC=C5)=N3)CCO2
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Shipping
Room temperature in continental US; may vary elsewhere.
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Storage
Please store the product under the recommended conditions in the Certificate of Analysis.
Purity & Documentation
References
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)
CYP121A1-IN-1 Related Classifications
HY-144325 Related Classifications
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