3083307-47-2
Chemical Structure
(R)-AR/BRD4 RIPTAC-1
- CAS No.: 3083307-47-2
- Formula:C50H54N10O5S
- Molecular Weight:907.09
InChIKey: PVYWAVIGWFSXIT-BMWAMRAGSA-N
SMILES: N#CC1=C(OC)C=C(O[C@@H]2C(C)(C)[C@@H](NC(C3=CN=C(N4CCC5(CC(OC6=CC=C(C7=N[C@H](CC8=NC=CO8)C9=NN=C(C)N9C%10=C7C(C)=C(C)S%10)C=C6)C5)CC4)N=C3)=O)C2(C)C)C=C1
Biological Activity: (R)-AR/BRD4 RIPTAC-1 is the R-enantiomer of AR/BRD4 RIPTAC-1 (HY-176521). AR/BRD4 RIPTAC-1 is an orally active Regulated Induced Proximity TArgeting Chimera (RIPTAC). AR/BRD4 RIPTAC-1 induces the formation of a stable ternary complex between the androgen receptor (AR) and BRD4, thereby blocking BRD4 function. AR/BRD4 RIPTAC-1 inhibits the growth and proliferation of tumor cells. AR/BRD4 RIPTAC-1 holds promise for research into prostate cancer.
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(R)-AR/BRD4 RIPTAC-1 | (R)-AR/BRD4 RIPTAC-1 is the R-enantiomer of AR/BRD4 RIPTAC-1 (HY-176521). AR/BRD4 RIPTAC-1 is an orally active Regulated Induced Proximity TArgeting Chimera (RIPTAC). AR/BRD4 RIPTAC-1 induces the formation of a stable ternary complex between the androgen receptor (AR) and BRD4, thereby blocking BRD4 function. AR/BRD4 RIPTAC-1 inhibits the growth and proliferation of tumor cells. AR/BRD4 RIPTAC-1 holds promise for research into prostate cancer. | |||||||||||||||||||||
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