873327-59-4
873327-59-4
Chemical Structure
AR-C141990
- CAS No.: 873327-59-4
- Formula:C26H28N4O4S
- Molecular Weight:492.59
IUPAC Name: (R)-5-(3-hydroxypyrrolidine-1-carbonyl)-1-isobutyl-3-methyl-6-(quinolin-4-ylmethyl)thieno[2,3-d]pyrimidine-2,4(1H,3H)-dione
InChIKey: JOFQERPJMGKMMX-QGZVFWFLSA-N
SMILES: O=C1N(CC(C)C)C2=C(C(C(N3C[C@H](O)CC3)=O)=C(CC4=CC=NC5=CC=CC=C45)S2)C(N1C)=O
Biological Activity: AR-C141990 (Compound 30) is a potent blocker of the monocarboxylate transporter MCT1 with a Ki of 4.8 nM. AR-C141990 (Compound 30) inhibits CYP3A4 and CYP2C9 with IC50 values of 16 μM[1].
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AR-C141990 | AR-C141990 (Compound 30) is a potent blocker of the monocarboxylate transporter MCT1 with a Ki of 4.8 nM. AR-C141990 (Compound 30) inhibits CYP3A4 and CYP2C9 with IC50 values of 16 μM. | |||||||||||||||||||||
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References
Keywords
