873336-87-9
Chemical Structure
Muscarinic toxin 3
Synonym(s): MT3
- CAS No.: 873336-87-9
- Formula:C319H489N89O97S8
- Molecular Weight:7379.35
SMILES: O=C([C@@H](N)CC(C)C)N[C@H](C(N[C@H](C(N[C@H](C(N[C@H](C(N[C@H](C(N[C@H](C(N[C@H](C(N[C@H](C(N[C@H](C(NCC(N[C@H](C(N[C@H](C(N[C@H](C(N[C@H](C(N[C@H](C(N[C@H](C(N1C(C(NC(C(NCC(NC(C(NC(C(NC2CC(C)C)=O)CC(N)=O)=O)CCC(N)=O)=O)=O)C)=O)CCC1)=O)CSSC[C@H](N3)C(N[C@H](C(N[C@H](C(N[C@H](C(N[C@H](C(N4[C@H](C(N[C@H](C(N5[C@H](C(N[C@H](C(N[C@H](C(N[C@H](C(N[C@H](C(N[C@H](C(N[C@H](C(N[C@H]6CC7=CNC=N7)=O)[C@H](CC)C)=O)CO)=O)CC(O)=O)=O)CC8=CC=C(O)C=C8)=O)CC(N)=O)=O)CCC(O)=O)=O)CCC5)=O)[C@H](CC)C)=O)CCC4)=O)CSSC[C@H](NC6=O)C(N[C@H](C(N[C@H](C(N[C@H](C(N[C@H](C(N[C@H]9CCCCN)=O)CC(O)=O)=O)[C@@H](C)O)=O)CCCCN)=O)CSSC[C@H](NC9=O)C(N[C@H](C(N[C@H](C(O)=O)CCC(O)=O)=O)CC(N)=O)=O)=O)=O)[C@@H](C)O)=O)C)=O)C)=O)=O)CC(N)=O)=O)CCC(O)=O)=O)[C@@H](C)O)=O)[C@@H](C)O)=O)[C@H](CC)C)=O)=O)CC%10=CC=CC=C%10)=O)[C@H](CC)C)=O)[C@@H](C)O)=O)CC(N)=O)=O)CCCCN)=O)[C@@H](C)O)=O)C(C)C)=O)CSSC[C@H](NC2=O)C(N[C@H](C(N[C@H](C(N[C@H](C(N[C@H](C(N[C@H](C(N[C@H](C(N[C@H](C(N[C@H](C(N%11[C@H](C(N[C@H](C(N[C@H](C(N[C@H](C(N[C@H](C(N[C@H](C(N[C@H](C(N[C@H](C(NCC3=O)=O)CCCNC(N)=N)=O)[C@@H](C)O)=O)[C@H](CC)C)=O)CCC(O)=O)=O)[C@@H](C)O)=O)CC%12=CC=C(O)C=C%12)=O)CCCNC(N)=N)=O)CCC%11)=O)[C@H](CC)C)=O)C(C)C)=O)CC%13=CC=C(O)C=C%13)=O)CC%14=CNC=N%14)=O)CC%15=CNC%16=CC=CC=C%15%16)=O)CCCNC(N)=N)=O)CCCCN)=O)CC%17=CC=CC=C%17)=O)=O)[C@@H](C)O
Biological Activity: Muscarinic toxin 3 (MT3) is a potent and non-competitive mAChR and adrenoceptors antagonist with pIC50s of 6.71, 8.79, 8.86, 7.57, 8.13, 8.49, <6.5, 7.29 against M1, M4, α1A, α1B, α1D,α2A,α2B and α2C receptors, respectively. Muscarinic toxin 3 displays prominent adrenoceptor activity[1].
| Cat. No. | Product Name | Purity | Description | Pricing | |||||||||||||||||||
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Muscarinic toxin 3 | Muscarinic toxin 3 (MT3) is a potent and non-competitive mAChR and adrenoceptors antagonist with pIC50s of 6.71, 8.79, 8.86, 7.57, 8.13, 8.49, <6.5, 7.29 against M1, M4, α1A, α1B, α1D,α2A,α2B and α2C receptors, respectively. Muscarinic toxin 3 displays prominent adrenoceptor activity. | |||||||||||||||||||||
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Keywords
