959705-64-7
959705-64-7
Chemical Structure
TC-E 5005
- CAS No.: 959705-64-7
- Formula:C15H18N4O
- Molecular Weight:270.33
IUPAC Name: 2-methoxy-6,7-dimethyl-9-propylimidazo[1,5-a]pyrido[3,2-e]pyrazine
InChIKey: YNADXFWEXJTQSZ-UHFFFAOYSA-N
SMILES: COC1=CC=C2C(N3C(C(C)=N2)=C(C)N=C3CCC)=N1
Biological Activity: TC-E 5005 is a potent and selective PDE10A inhibitor with IC50 values of 7.28, 239, 779, 919, 3,100, and 3,700 nM for PDE10A, 2A, 11A, 5A, 7B and 3A, respectively. TC-E 5005 inhibits adrenergic and neurogenic smooth muscle contractions in the human prostate[1].
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TC-E 5005 | TC-E 5005 is a potent and selective PDE10A inhibitor with IC50 values of 7.28, 239, 779, 919, 3,100, and 3,700 nM for PDE10A, 2A, 11A, 5A, 7B and 3A, respectively. TC-E 5005 inhibits adrenergic and neurogenic smooth muscle contractions in the human prostate. | |||||||||||||||||||||
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References
Keywords
