BRL-41992
BRL-41992 is a selective α₂B-adrenergic receptor antagonist. BRL-41992 exhibits 94-fold higher selectivity for the α₂B-receptor than for the α₂A-receptor with Kᵢ values in neonatal rat lung tissue (expressing the α₂B-receptor) and in human platelet membranes (expressing the α₂A-receptor) of 1.1 and 103.3 nM. BRL-41992 can be used to verify the functional differences of α₂ receptor subtypes.
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- CAS No.: 124097-52-5
- Formule: C18H20N2
- Masse moléculaire:264.36
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Stockage:
Please store the product under the recommended conditions in the Certificate of Analysis.
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Activité biologique
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Chemical Information
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Activité biologique
Description
IC50 & Target
[1]|
Alpha-2A adrenergic receptor 1.1 nM (Ki) |
Alpha-2B adrenergic receptor 103.3 nM (Ki) |
Chemical Information
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CAS No. 124097-52-5
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Masse moléculaire 264.36
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Formule C18H20N2
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SMILES
CN(CN1[C@]2(C3=CC=CC=C3CC4=CC=CC=C41)[H])[C@@H]2C
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Livraison
Room temperature in continental US; may vary elsewhere.
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Stockage
Please store the product under the recommended conditions in the Certificate of Analysis.
Pureté et documentation
Références
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)
BRL-41992 Related Classifications
HY-118200 Related Classifications
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