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CP-100356

9 Cited Publications
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Based on 9 publication(s) in Google Scholar

CP-100356 is an orally active dual MDR1 (P-gp)/BCRP inhibitor, with an IC50s of 0.5 and 1.5 µM for inhibiting MDR1-mediated Calcein-AM transport and BCRP-mediated Prazosin transport, respectively. CP-100356 is also a weak inhibitor of OATP1B1 (IC50 = ∼66 µM). CP-100356 is devoid of inhibition against MRP2 and major human P450 enzymes (IC50 > 15 µM).

For research use only. We do not sell to patients.

  • CAS No.: 142716-85-6
  • Formula: C31H36N4O6
  • Molecular Weight:560.64
  • Storage:

    Please store the product under the recommended conditions in the Certificate of Analysis.

  • CP-100356 Chemical Structure
    CP-100356 Chemical Structure
CAS No.: 142716-85-6
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609-228-6898
[email protected] [email protected]
Find Your Local Distributor Your local distributor: Hycultec GmbHHycultec
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Publications Citing Use of MedChemExpress (MCE) CP-100356

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    CP-100356 Chemical Structure
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