2. Metabolic Enzyme/Protease
  3. Cytochrome P450
  4. CYP3A4-IN-2

CYP3A4-IN-2 is a specific inhibitor of cytochrome P450 3A4 (CYP3A4) with the IC50 value of 0.055 μM. CYP3A4-IN-2 is a ritonavir analogue with increased hydrophobicity of the R2 side group and stronger inhibitory effect compared to ritonavir. CYP3A4-IN-2 can be used as an antiviral agent and immunosuppressants.

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CYP3A4-IN-2

CYP3A4-IN-2 Chemical Structure

CAS No. : 2562383-94-0

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CYP3A4-IN-2 Related Antibodies

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Voir tous les produits spécifiques à Isoform Cytochrome P450:

Voir toutes les isoformes
CYP1 CYP2 CYP3 CYP4 CYP11 CYP17 Aromatase/CYP19A1 CYP26 CYP51 CYP1A2 CYP2D6 CYP2C9 CYP2C19 CYP3A CYP3A4 CYP17A1

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Description

CYP3A4-IN-2 is a specific inhibitor of cytochrome P450 3A4 (CYP3A4) with the IC50 value of 0.055 μM. CYP3A4-IN-2 is a ritonavir analogue with increased hydrophobicity of the R2 side group and stronger inhibitory effect compared to ritonavir. CYP3A4-IN-2 can be used as an antiviral agent and immunosuppressants[1].

IC50 & Target

CYP3A4

0.055 μM (IC50)

Masse moléculaire

570.74

Formule

C33H38N4O3S
CAS No.
SMILES

O=C(OC(C)(C)C)NC(CC1=C2C=CC=CC2=CC=C1)CSCC(NC3=CC=CC=C3)C(NCC4=CC=CN=C4)=O
Livraison

Room temperature in continental US; may vary elsewhere.
Stockage

Please store the product under the recommended conditions in the Certificate of Analysis.
Pureté et documentation
Références
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CYP3A4-IN-2 Related Classifications

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The dilution calculator equation

Concentration (start) × Volume (start) = Concentration (final) × Volume (final)

This equation is commonly abbreviated as: C1V1 = C2V2

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× = ×
C1   V1   C2   V2
Help & FAQs
  • Do most proteins show cross-species activity?

    Species cross-reactivity must be investigated individually for each product. Many human cytokines will produce a nice response in mouse cell lines, and many mouse proteins will show activity on human cells. Other proteins may have a lower specific activity when used in the opposite species.

Keywords:

CYP3A4-IN-22562383-94-0Cytochrome P450CYPsCYP3A4 inhibitorritonavirantiviral agentimmunosuppressantInhibitorinhibitorinhibit

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