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Cat. No.: HY-102092

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FR139317

Name: FR139317
Brand: MedChemExpress
SKU: HY-102092
Availability: PreOrder

(Synonyms: PD 147953)

FR139317 (PD 147953) is a selective ET_A receptor antagonist. FR139317 inhibits cerebral activation by intraventricular endothelin-1 in conscious rats. FR139317 also ameliorates cerebral vasospasm in dogs.

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CAS No.: 142375-60-8
화학식: C₃₃H₄₄N₆O₅
분자량:604.74

보관:

Please store the product under the recommended conditions in the Certificate of Analysis.

Data Sheet (271 KB)

FR139317 Chemical Structure

CAS No.: 142375-60-8

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^[1]

ET_A

All Endothelin Receptor Isoforms :

ET_A
ET_B

Chemical Information

CAS No. 142375-60-8
분자량 604.74
화학식 C₃₃H₄₄N₆O₅
SMILES

O=C(O)[C@@H](CC1=NC=CC=C1)NC([C@@H](CC2=CN(C)C3=CC=CC=C23)NC([C@H](CC(C)C)NC(N4CCCCCC4)=O)=O)=O
Synonyms

PD 147953
선적

Room temperature in continental US; may vary elsewhere.
보관

Please store the product under the recommended conditions in the Certificate of Analysis.

순도&문서

Select Batch:

Purity: 99.98%

Assay: 99.98%

ee.: 99.98%

Data Sheet (271 KB)
COA (2659 KB)
Elemental Analysis Report (2659 KB)
HNMR (2659 KB)
CNMR (2659 KB)
RP-HPLC (2659 KB)
NP-HPLC (2659 KB)
MS (2659 KB)
LCMS (2659 KB)
IR (2659 KB)
GC (2659 KB)
OR (2659 KB)
SDS-PAGE (2659 KB)
SEC-HPLC (2659 KB)
Other Report (2659 KB)
Handling Instructions (2659 KB)

References

[1]. Gross PM, et al. FR139317, a specific ETA-receptor antagonist, inhibits cerebral activation by intraventricular endothelin-1 in conscious rats. Neuropharmacology. 1994 Oct;33(10):1155-66. [Content Brief]

[2]. Nirei H, et al. An endothelin ETA receptor antagonist, FR139317, ameliorates cerebral vasospasm in dogs. Life Sci. 1993;52(23):1869-74. [Content Brief]

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How should lyophilized recombinant proteins be reconstituted and stored?

1. Before opening the cap, centrifuge the vial at 13000 rpm for 20-30 seconds. This step will ensure that any lyophilized powder that may have adhered to the cap or walls is collected at the bottom of the vial, minimizing the risk of product loss.

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FR139317

All Endothelin Receptor Isoforms

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