1. Cell Cycle/DNA Damage
    Epigenetics
  2. PARP
    Histone Methyltransferase
  3. PARP/EZH2-IN-1

PARP/EZH2-IN-1 

Cat. No.: HY-132885
Handling Instructions

PARP/EZH2-IN-1 is a first-in-class dual PARP (IC50 6.87 nM) and EZH2 (IC50 36.51 nM) inhibitor for triple-negative breast cancer with wild-type BRCA.

For research use only. We do not sell to patients.

PARP/EZH2-IN-1 Chemical Structure

PARP/EZH2-IN-1 Chemical Structure

CAS No. : 2687273-52-3

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Description

PARP/EZH2-IN-1 is a first-in-class dual PARP (IC50 6.87 nM) and EZH2 (IC50 36.51 nM) inhibitor for triple-negative breast cancer with wild-type BRCA.

IC50 & Target

PARP-1

6.87 nM (IC50)

EZH2

36.51 nM (IC50)

Molecular Weight

768.83

Formula

C₄₃H₄₁FN₈O₅

CAS No.
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Storage

Please store the product under the recommended conditions in the Certificate of Analysis.

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Product Name:
PARP/EZH2-IN-1
Cat. No.:
HY-132885
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