1. PROTAC
  2. E3 Ligase Ligand-Linker Conjugates
  3. (S,R,S)-AHPC-Me-C5-COOH

(S,R,S)-AHPC-Me-C5-COOH 

Cat. No.: HY-130849 Purity: 96.19%
Handling Instructions

(S,R,S)-AHPC-Me-C5-COOH is a synthesized E3 ligase ligand-linker conjugate that incorporates the a VHL ligand and a linker. (S,R,S)-AHPC-Me-C5-COOH can be used in PROTAC DT2216 (HY-130604).

For research use only. We do not sell to patients.

(S,R,S)-AHPC-Me-C5-COOH Chemical Structure

(S,R,S)-AHPC-Me-C5-COOH Chemical Structure

CAS No. : 2229976-21-8

Size Price Stock Quantity
50 mg USD 960 In-stock
Estimated Time of Arrival: December 31
100 mg USD 1550 In-stock
Estimated Time of Arrival: December 31
200 mg   Get quote  
500 mg   Get quote  

* Please select Quantity before adding items.

Customer Review

Based on 1 publication(s) in Google Scholar

Top Publications Citing Use of Products

View All E3 Ligase Ligand-Linker Conjugates Isoform Specific Products:

  • Biological Activity

  • Purity & Documentation

  • References

  • Customer Review

Description

(S,R,S)-AHPC-Me-C5-COOH is a synthesized E3 ligase ligand-linker conjugate that incorporates the a VHL ligand and a linker. (S,R,S)-AHPC-Me-C5-COOH can be used in PROTAC DT2216 (HY-130604)[1].

IC50 & Target[1]

VHL

 

In Vitro

DT2216 is a selective B-cell lymphoma extra large (BCL-XL) PROTAC degrader[1].

MCE has not independently confirmed the accuracy of these methods. They are for reference only.

Molecular Weight

586.74

Formula

C30H42N4O6S

CAS No.
SMILES

O=C(N[[email protected]](C1=CC=C(C2=C(C)N=CS2)C=C1)C)[[email protected]]3N(C([[email protected]](C(C)(C)C)NC(CCCCCC(O)=O)=O)=O)C[[email protected]](O)C3

Shipping

Room temperature in continental US; may vary elsewhere.

Storage

4°C, sealed storage, away from moisture

*In solvent : -80°C, 6 months; -20°C, 1 month (sealed storage, away from moisture)

References
  • No file chosen (Maximum size is: 1024 Kb)
  • If you have published this work, please enter the PubMed ID.
  • Your name will appear on the site.
  • Molarity Calculator

  • Dilution Calculator

The molarity calculator equation

Mass (g) = Concentration (mol/L) × Volume (L) × Molecular Weight (g/mol)

Mass   Concentration   Volume   Molecular Weight *
= × ×

The dilution calculator equation

Concentration (start) × Volume (start) = Concentration (final) × Volume (final)

This equation is commonly abbreviated as: C1V1 = C2V2

Concentration (start) × Volume (start) = Concentration (final) × Volume (final)
× = ×
C1   V1   C2   V2

Your Recently Viewed Products:

Inquiry Online

Your information is safe with us. * Required Fields.

Product Name

 

Salutation

Applicant Name *

 

Email address *

Phone number *

 

Organization name *

Department *

 

Requested quantity *

Country or Region *

     

Remarks

Bulk Inquiry

Inquiry Information

Product Name:
(S,R,S)-AHPC-Me-C5-COOH
Cat. No.:
HY-130849
Quantity:
MCE Japan Authorized Agent: