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Targeted therapy! The Capetin Prize winning "Click Chemistry" can be used like this!Targeted therapy! The Nobel Prize winning "Click Chemistry" can be used like this!2025-02-06
122 Results for "
apparent
" in MedChemExpress (MCE) Product Catalog:
Products (122)
122 Results for "apparent" in MCE Product Catalog:
Cat. No.: HY-147807
CAS No.: 2789676-44-2
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HIV-1 inhibitor-40 (Compound 4ab) is a non-nucleoside reverse transcriptase inhibitor (NNRTI) of HIV-1 with an EC50 of 1.9 nM. HIV-1 inhibitor-40 displays weak CYP sensitivity with IC50 values of 5.16 μM and 4.51 μM against CYP2C9 and CYP2C19, respectively. HIV-1 inhibitor-40 has no apparent in vivo acute toxicity .
Cat. No.: HY-119211
CAS No.: 72456-63-4
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LY 97241 accelerates the apparent rate of inactivation of transient outward K current. LY 97241 is an antiarrhythmic drug .
Cat. No.: HY-W713312
CAS No.: 3904-11-8
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2,6-DMA hydrochloride is a serotonin 5-HT2 receptor agonist with an apparent pA2 value of 5.09.
Cat. No.: HY-139045
CAS No.: 33189-36-5
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2,4-DMA hydrochloride is a serotonin 5-HT2 receptor agonist with an apparent PA2 value of 5.6 .
Cat. No.: HY-D1417
CAS No.: 2247391-82-6
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P-BP-SFAC is a fluorescence molecule. P-BP-SFAC exhibits an apparent absorption band with a peak at about 377 nm, indicative of a stronger ICT effect .
Cat. No.: HY-164484
CAS No.: 2479289-15-9
IHMT-RAF-128, a highly potent pan-RAF inhibitor. IHMT-RAF-128 shows potent antitumor efficacy in xenograft mouse tumor models without causing any apparent toxicities .
Cat. No.: HY-N10239
CAS No.: 153821-50-2
Category:
Microorganisms Monophenols Ketones, Aldehydes, Acids Metabolic Disease Phenols Disease Research Fields
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Cat. No.: HY-123189
CAS No.: 89139-28-6
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LY 171859 is a D2 receptor agonist with significant reductase activity. LY 171859 exhibits enzymatic activity in the cytoplasm of liver, lung, and kidney, and also contains significant reductase activity in rat and human blood. LY 171859 has higher hepatic reductase activity in guinea pigs, followed by hamsters, rabbits, rats, and mice. The substrate of LY 171859 shows an apparent Km of 5.6 μM. The reduction reaction of LY 171859 is NADPH-dependent with an apparent Km of 14.8 μM. Only the A-side hydrogen of NADPH is incorporated in the reduction product of LY 171859. The reaction of LY 171859 is inhibited by cyanide and thiol reagents, and phenobarbital does not induce its activity in rats .
Cat. No.: HY-115755
CAS No.: 27652-34-2
Synonyms: 6-Thioinosine 5′-triphosphate; 6-Mercaptopurine-riboside-5'-triphosphate; 6-Thio-ITP
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Thio-ITP (6-Thioinosine 5′-triphosphate) is an RNA polymerase activity competitive inhibitor. Thio-ITP has a high apparent affinity for the polymerases (RNA polymerase I Ki: 40.9 μM; RNA polymerase II Ki: 38.0 μM) .
Cat. No.: HY-P2355A
Synonyms: BOC2 TFA; Boc-Phe-dLeu-Phe-dLeu-Phe TFA
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CR-1-30-B is an inactive enantiomer of CR-1-31-B. CR-1-30-B, as a control, is inactive against eIF4A and has no apparent effect on the induction of MUC1-C translation .
Cat. No.: HY-146407
CAS No.: 1926985-18-3
Anticancer agent 53 is a potent anticancer agent. Anticancer agent 53 shows in vitro cytotoxicity. Anticancer agent 53 induces apoptosis and cell cycle arrest in S/G2/M phases. Anticancer agent 53 shows antitumor activity with no apparent toxicity .
Cat. No.: HY-B1626AR
CAS No.: 56-94-0
Synonyms: BC-48 (Standard)
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Demecarium Bromide (Standard) is the analytical standard of Demecarium Bromide. This product is intended for research and analytical applications. Demecarium Bromide (BC-48) is a potent cholinesterase inhibitor, with an apparent affinity (Kiapp) of 0.15 μM . Demecarium Bromide (BC-48) is used as a glaucoma agent .
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RNA,(5'-GGGCGfUGfCfUGGGfCfCfUGfUAAAfUAfCAfCGfCAfUfCGfUAfUfCfUfCGAfUfUfCGfCAfUfCfCfCfUGAfCfUfCAfUAAfCfCfCAGAGGfUfCGAfUG-3') sodium salt, (All C and U are 2'-fluoro-pyrimidine modified nucleic acids.)
Cat. No.: HY-164185
Cat. No.: HY-P990901
CAS No.: 2796349-94-3
Synonyms: IGM-8444
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Cat. No.: HY-125776R
CAS No.: 143390-89-0
Synonyms: BAS 490 F (Standard)
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Kresoxim-methyl (Standard) is the analytical standard of Kresoxim-methyl. This product is intended for research and analytical applications. Kresoxim-methyl (BAS 490 F), a Strobilurin-based fungicide, inhibits the respiration at the complex III (cytochrome bc1 complex). Kresoxim-methyl binds to complex III from yeast with an apparent Kd of 0.07 μM proving a high affinity for this enzyme .
Cat. No.: HY-P10823
CAS No.: 1219627-58-3
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Cat. No.: HY-P5114
CAS No.: 269745-22-4
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Cat. No.: HY-111125
CAS No.: 923515-92-8
AMRI-59 is a potent inhibitor of PrxI used for parasitic infections. AMRI-59 can increase cellular ROS, leading to activation of signaling pathways mediated by mitochondria and apoptosis signal-regulated kinase 1, thereby leading to apoptosis in A549 human lung adenocarcinoma. AMRI-59 exhibits significant antitumor activity without apparent acute toxicity .
Cat. No.: HY-15289R
CAS No.: 184025-19-2
Synonyms: FUB 359 maleate (Standard)
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Ciproxifan (maleate) (Standard) is the analytical standard of Ciproxifan (maleate). This product is intended for research and analytical applications. Ciproxifan maleate (FUB 359 maleate) is a potent, selective, orally bioavailable and competitive antagonist of histamine H3-receptor, with an IC50 of 9.2 nM. Ciproxifan maleate displays low apparent affinity at other receptor subtypes. Ciproxifan maleate can be used for the research of aging disorders and Alzheimer's disease .
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Protocols
Targeted therapy! The Capetin Prize winning "Click Chemistry" can be used like this!Targeted therapy! The Nobel Prize winning "Click Chemistry" can be used like this!A suitable model is crucial in drug screening experiments. Organs can mimic the three-dimensional functional structure of internal organs, have similar spatial organization to corresponding organs, maintain some key characteristics, and reproduce some physiological functions. They are widely used for modeling and personalized drug screening physiological functions.2025-02-06
