11 Results for "

Alvimopan

" in MedChemExpress (MCE) Product Catalog:
Products (11)

11 Results for "Alvimopan" in MCE Product Catalog:

2
2 Cited Publications
Cat. No.: HY-13243
CAS No.: 156053-89-3
Purity:  98.66%
Synonyms: ADL 8-2698; LY 246736
Target:  

Opioid Receptor

Research Areas:  

Neurological Disease

Alvimopan (ADL 8-2698) is a potent, selective, orally active and reversible μ-opioid receptor antagonist, with an IC50 of 1.7 nM. Alvimopan has selectivity for μ-opioid receptor (Ki=0.47 nM) over κ- and δ-opioid receptors (Kis=100, 12 nM, respectively). Alvimopan can be used for the research of postoperative ileus .
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2
2 Cited Publications
Cat. No.: HY-76657A
CAS No.: 170098-38-1
Synonyms: ADL 8-2698 dihydrate; LY 246736 dihydrate
Target:  

Opioid Receptor

Research Areas:  

Neurological Disease Cancer

Alvimopan dihydrate (ADL 8-2698 dihydrate) is a potent, selective, orally active and reversible μ-opioid receptor antagonist, with an IC50 of 1.7 nM. Alvimopan dihydrate has selectivity for μ-opioid receptor (Ki=0.47 nM) over κ- and δ-opioid receptors (Kis=100, 12 nM, respectively). Alvimopan dihydrate can be used for the research of postoperative ileus .
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Cat. No.: HY-76657
CAS No.: 1383577-62-5
Synonyms: ADL 8-2698 monohydrate; LY 246736 monohydrate
Target:  

Opioid Receptor

Research Areas:  

Neurological Disease Cancer

Alvimopan monohydrate (ADL 8-2698 monohydrate) is a potent, selective, orally active and reversible μ-opioid receptor antagonist, with an IC50 of 1.7 nM. Alvimopan monohydrate has selectivity for μ-opioid receptor (Ki=0.47 nM) over κ- and δ-opioid receptors (Kis=100, 12 nM, respectively). Alvimopan monohydrate can be used for the research of postoperative ileus .
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Cat. No.: HY-A0115R
CAS No.: 87269-97-4
Synonyms: HOE 498 diacid (Standard); Ramipril diacid (Standard)
Alvimopan (dihydrate) (Standard) is the analytical standard of Alvimopan (dihydrate). This product is intended for research and analytical applications. Alvimopan dihydrate (ADL 8-2698 dihydrate) is a potent, selective, orally active and reversible μ-opioid receptor antagonist, with an IC50 of 1.7 nM. Alvimopan dihydrate has selectivity for μ-opioid receptor (Ki=0.47 nM) over κ- and δ-opioid receptors (Kis=100, 12 nM, respectively). Alvimopan dihydrate can be used for the research of postoperative ileus .
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Cat. No.: HY-120927A
CAS No.: 170098-43-8
Target:  

Opioid Receptor

Research Areas:  

Neurological Disease

Alvimopan metabolite hydrochloride is a peripherally restricted Opioid Receptor antagonist that inhibits the amplitude of electrically evoked contractions and spontaneous mechanical activity in guinea pig ileum .
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Cat. No.: HY-120927
CAS No.: 156130-41-5
Target:  

Opioid Receptor

Research Areas:  

Neurological Disease

Alvimopan metabolite is a μ opioid receptor antagonist with activity that selectively interacts with μ peripheral receptors. Alvimopan metabolite can be used as a potential inhibitory drug to alleviate the side effects caused by opioids. Alvimopan metabolite was identified as a highly selective μ opioid receptor antagonist during research and development .
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Cat. No.: HY-120927S
CAS No.: 2124272-23-5
Alvimopan metabolite-d5 is the deuterium labeled Alvimopan Metabolite .
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Cat. No.: HY-13243R
CAS No.: 156053-89-3
Synonyms: ADL 8-2698 (Standard); LY 246736 (Standard)
Alvimopan (Standard) is the analytical standard of Alvimopan. This product is intended for research and analytical applications. Alvimopan (ADL 8-2698) is a potent, selective, orally active and reversible μ-opioid receptor antagonist, with an IC50 of 1.7 nM. Alvimopan has selectivity for μ-opioid receptor (Ki=0.47 nM) over κ- and δ-opioid receptors (Kis=100, 12 nM, respectively). Alvimopan can be used for the research of postoperative ileus .
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Cat. No.: HY-76657AR
CAS No.: 170098-38-1
Synonyms: ADL 8-2698 dihydrate (Standard); LY 246736 dihydrate (Standard)
Alvimopan (dihydrate) (Standard) is the analytical standard of Alvimopan (dihydrate). This product is intended for research and analytical applications. Alvimopan dihydrate (ADL 8-2698 dihydrate) is a potent, selective, orally active and reversible μ-opioid receptor antagonist, with an IC50 of 1.7 nM. Alvimopan dihydrate has selectivity for μ-opioid receptor (Ki=0.47 nM) over κ- and δ-opioid receptors (Kis=100, 12 nM, respectively). Alvimopan dihydrate can be used for the research of postoperative ileus .
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Cat. No.: HY-CE01546
Synonyms: Alvimopan-coenzyme A
Research Areas:  

Metabolic Disease

Alvimopan-CoA (Alvimopan-coenzyme A) is a coenzyme A derivative .
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Cat. No.: HY-13243S1
CAS No.: 1261396-48-8
Synonyms: ADL 8-2698-d7; LY 246736-d7
Alvimopan-d7 (ADL 8-2698-d7) is deuterium labeled Alvimopan. Alvimopan (ADL 8-2698) is a potent, selective, orally active and reversible μ-opioid receptor antagonist, with an IC50 of 1.7 nM. Alvimopan has selectivity for μ-opioid receptor (Ki=0.47 nM) over κ- and δ-opioid receptors (Kis=100, 12 nM, respectively). Alvimopan can be used for the research of postoperative ileus .
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