7 Results for "

DS5565

" in MedChemExpress (MCE) Product Catalog:
Products (7)

7 Results for "DS5565" in MCE Product Catalog:

6
6 Cited Publications
Cat. No.: HY-12650
CAS No.: 1138245-13-2
Purity:  99.31%
Synonyms: DS5565
Target:  

Calcium Channel

Research Areas:  

Neurological Disease

Mirogabalin (DS-5565) is a novel, preferentially selective α2δ-1 ligand characterized by high potency and selectivity to the α2δ-1 subunit of voltage-sensitive calcium channel complexes in the CNS.
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6
6 Cited Publications
Cat. No.: HY-108006
CAS No.: 1138245-21-2
Purity:  99.57%
Synonyms: DS 5565 besylate
Target:  

Calcium Channel

Research Areas:  

Neurological Disease

Mirogabalin besylate is a selective and orally available ligand for the α2δ subunit of voltage-gated calcium channels, with Kds of 13.5 nM, 22.7 nM, 27 nM, and 47.6 nM for human α2δ-1, human α2δ-2, rat α2δ-1, and rat α2δ-2, respectively.
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Cat. No.: HY-12650S1
Synonyms: DS5565-d4
Mirogabalin-d4 (DS5565-d4) is a deuterated compound of Mirogabalin (HY-12650), a ligand that selectively targets the voltage-sensitive calcium channel complex α2δ-1 .
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Cat. No.: HY-12650R
CAS No.: 1138245-13-2
Synonyms: DS5565 (Standard)
Research Areas:  

Neurological Disease

Mirogabalin (Standard) is the analytical standard of Mirogabalin. This product is intended for research and analytical applications. Mirogabalin (DS-5565) is a novel, preferentially selective α2δ-1 ligand characterized by high potency and selectivity to the α2δ-1 subunit of voltage-sensitive calcium channel complexes in the CNS.
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Cat. No.: HY-12650S
Synonyms: DS5565-13C2,d1 (Mixture of Diastereomers)
Mirogabalin- 13C2,d1 (Mixture of Diastereomers) is a 13C and deuterium labeled Mirogabalin. Mirogabalin (DS-5565) is a preferentially selective α2δ-1 ligand characterized by high potency and selectivity to the α2δ-1 subunit of voltage-sensitive calcium channel complexes in the CNS .
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Cat. No.: HY-12650A
CAS No.: 1138244-97-9
Synonyms: (rel)-DS5565
Target:  

Calcium Channel

Research Areas:  

Neurological Disease

(rel)-Mirogabalin ((rel)-DS5565) is a voltage-dependent calcium channel inhibitor that acts on the α2δ-1 subunit .
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Cat. No.: HY-108006R
CAS No.: 1138245-21-2
Synonyms: DS 5565 besylate (Standard)
Research Areas:  

Neurological Disease

Mirogabalin besylate (Standard) is the analytical standard of Mirogabalin besylate (HY-108006). This product is intended for research and analytical applications. Mirogabalin besylate is a selective and orally available ligand for the α2δ subunit of voltage-gated calcium channels, with Kds of 13.5 nM, 22.7 nM, 27 nM, and 47.6 nM for human α2δ-1, human α2δ-2, rat α2δ-1, and rat α2δ-2, respectively.
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