1138245-21-2
1138245-21-2
Chemical Structure
Mirogabalin besylate
Synonym(s): DS 5565 besylate
- CAS No.: 1138245-21-2
- Formula:C18H25NO5S
- Molecular Weight:367.46
IUPAC Name: 2-((1R,5S,6S)-6-(aminomethyl)-3-ethylbicyclo[3.2.0]hept-3-en-6-yl)acetic acid compound with benzenesulfonic acid (1:1)
InChIKey: OKJXJRVWXYRSAN-TXULWXBWSA-N
SMILES: O=S(C1=CC=CC=C1)(O)=O.OC(C[C@@]2([C@@]3([H])[C@@](CC(CC)=C3)([H])C2)CN)=O
Biological Activity: Mirogabalin besylate is a selective and orally available ligand for the α2δ subunit of voltage-gated calcium channels, with Kds of 13.5 nM, 22.7 nM, 27 nM, and 47.6 nM for human α2δ-1, human α2δ-2, rat α2δ-1, and rat α2δ-2, respectively.
| Cat. No. | Product Name | Purity | Description | Pricing | |||||||||||||||||||
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Mirogabalin besylate | 99.57% | Mirogabalin besylate is a selective and orally available ligand for the α2δ subunit of voltage-gated calcium channels, with Kds of 13.5 nM, 22.7 nM, 27 nM, and 47.6 nM for human α2δ-1, human α2δ-2, rat α2δ-1, and rat α2δ-2, respectively. | ||||||||||||||||||||
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Mirogabalin besylate (Standard) | ≥98% | Mirogabalin besylate (Standard) is the analytical standard of Mirogabalin besylate (HY-108006). This product is intended for research and analytical applications. Mirogabalin besylate is a selective and orally available ligand for the α2δ subunit of voltage-gated calcium channels, with Kds of 13.5 nM, 22.7 nM, 27 nM, and 47.6 nM for human α2δ-1, human α2δ-2, rat α2δ-1, and rat α2δ-2, respectively. | ||||||||||||||||||||
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