1138245-13-2
1138245-13-2
Chemical Structure
Mirogabalin
Synonym(s): DS5565
- CAS. Nr.: 1138245-13-2
- Formula:C12H19NO2
- Molecular Weight:209.28
IUPAC Name: 2-((1R,5S,6S)-6-(aminomethyl)-3-ethylbicyclo[3.2.0]hept-3-en-6-yl)acetic acid
InChIKey: FTBQORVNHOIASH-CKYFFXLPSA-N
SMILES: O=C(O)C[C@]1(CN)[C@]2([H])C=C(CC)C[C@]2([H])C1
Biological Activity: Mirogabalin (DS-5565) is a novel, preferentially selective α2δ-1 ligand characterized by high potency and selectivity to the α2δ-1 subunit of voltage-sensitive calcium channel complexes in the CNS.
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Mirogabalin | 99.22% | Mirogabalin (DS-5565) is a novel, preferentially selective α2δ-1 ligand characterized by high potency and selectivity to the α2δ-1 subunit of voltage-sensitive calcium channel complexes in the CNS. | ||||||||||||||||||||
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Mirogabalin (Standard) | ≥98% | Mirogabalin (Standard) is the analytical standard of Mirogabalin. This product is intended for research and analytical applications. Mirogabalin (DS-5565) is a novel, preferentially selective α2δ-1 ligand characterized by high potency and selectivity to the α2δ-1 subunit of voltage-sensitive calcium channel complexes in the CNS. | ||||||||||||||||||||
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Mirogabalin-d4 | Mirogabalin-d4 (DS5565-d4) is a deuterated compound of Mirogabalin (HY-12650), a ligand that selectively targets the voltage-sensitive calcium channel complex α2δ-1. | |||||||||||||||||||||
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Mirogabalin-13C2,d1 (Mixture of Diastereomers) | Mirogabalin-13C2,d1 (Mixture of Diastereomers) is a 13C and deuterium labeled Mirogabalin. Mirogabalin (DS-5565) is a preferentially selective α2δ-1 ligand characterized by high potency and selectivity to the α2δ-1 subunit of voltage-sensitive calcium channel complexes in the CNS. | |||||||||||||||||||||
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Jasmonic acid | Jasmonic acid ((-)-Jasmonic acid) is a plant growth regulator and a derivative of Linolenic acid (HY-N0728). Jasmonic acid enhances plant resistance and is widely used as a stress protectant. Jasmonic acid is an endogenous plant hormone and a plant growth inhibitor. | |||||||||||||||||||||
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7-epi Jasmonic acid | 7-epi Jasmonic acid is the isomer of (±)-Jasmonic acid (HY-122464). (±)-Jasmonic acid is a plant growth regulator and a derivative of α-linolenic acid. (±)-Jasmonic acid decreases chlorophyll levels in green and etiolated barley leaf segments and inhibits elongation of rice seedlings. | |||||||||||||||||||||
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(rel)-Mirogabalin | (rel)-Mirogabalin ((rel)-DS5565) is a voltage-dependent calcium channel inhibitor that acts on the α2δ-1 subunit. | |||||||||||||||||||||
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PD-217014-methyl ester | PD-217014-methyl ester is an α?δ ligand with visceral analgesic activity and can inhibit visceral hypersensitivity, and its anti-hyperalgesic effect is dose-dependent. | |||||||||||||||||||||
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PD-217014 | PD-217014 is an α2δ ligand with visceral analgesic activity and can inhibit visceral hypersensitivity reactions. Its anti-allodynic effect is dose-dependent. | |||||||||||||||||||||
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Atagabalin | Atagabalin (PD 0200390) is a Voltage-gated Calcium channel α2δ subunit binder with an IC50 of 22 nM. Atagabalin regulates neurotransmitter release by inhibiting calcium influx at high neuronal firing rates. Atagabalin can be used in research related to sleep disorders. | |||||||||||||||||||||
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iso-Atagabalin hydrochloride | iso-Atagabalin (iso-PD 0200390) hydrochloride is a stereoisomer of Atagabalin (HY-14856). Atagabalin is a selective GABA (gamma-aminobutyric acid) receptor agonist with antianxiety effect. | |||||||||||||||||||||
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Atagabalin hydrochloride | Atagabalin hydrochloride (PD 0200390 hydrochloride) is a Voltage-gated Calcium channel α2δ subunit binder with an IC50 of 22 nM. Atagabalin hydrochloride regulates neurotransmitter release by inhibiting calcium influx at high neuronal firing rates. Atagabalin hydrochloride can be used in research related to sleep disorders. | |||||||||||||||||||||
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Gabapentin | 99.99% | Gabapentin is a potent, orally active P/Q type Ca2+ channel blocker. Gabapentin inhibits neuronal Ca2+ influx and reduction of neurotransmitter release. Gabapentin is a GABA analog that can be used to relieve neuropathic pain. | ||||||||||||||||||||
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(Rac)-Jasmonic acid | (Rac)-Jasmonic acid is the racemate of Jasmonic acid (HY-122464A). Jasmonic acid ((-)-Jasmonic acid) is a plant growth regulator and a derivative of Linolenic acid (HY-N0728). | |||||||||||||||||||||
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