8 Results for "

GDC0973

" in MedChemExpress (MCE) Product Catalog:
Products (8)

8 Results for "GDC0973" in MCE Product Catalog:

63
63 Cited Publications
Cat. No.: HY-13064
CAS No.: 934660-93-2
Purity:  99.81%
Synonyms: GDC-0973; XL518
Target:  

MEK Apoptosis

Research Areas:  

Cancer

Cobimetinib (GDC-0973, RG7420) is a potent, selective and oral MEK1 inhibitor with an IC50 of 4.2 nM for MEK1.
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63
63 Cited Publications
Cat. No.: HY-13064A
CAS No.: 1369665-02-0
Purity:  99.73%
Synonyms: GDC-0973 hemifumarate; XL-518 hemifumarate
Target:  

MEK Apoptosis

Research Areas:  

Cancer

Cobimetinib hemifumarate is a novel selective MEK1 inhibitor, and the IC50 value against MEK1 is 4.2 nM.
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Cat. No.: HY-13078
CAS No.: 934662-91-6
Purity:  99.39%
Synonyms: GDC-0973 racemate; XL518 racemate
Target:  

MEK

Research Areas:  

Cancer

Cobimetinib racemate (GDC-0973 racemate; XL518 racemate) is the racemate of Cobimetinib. Cobimetinib is a potent and selective MEK inhibitor.
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Cat. No.: HY-13064S1
Synonyms: GDC-0973-d4hydrochloride; XL518-d4 hydrochloride
Cobimetinib-d4 hydrochloride is deuterated labeled Cobimetinib (HY-13064). Cobimetinib (GDC-0973, RG7420) is a potent, selective and oral MEK1 inhibitor with an IC50 of 4.2 nM for MEK1.
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Cat. No.: HY-13064R
CAS No.: 934660-93-2
Synonyms: GDC-0973 (Standard); XL518 (Standard)
Research Areas:  

Cancer

Cobimetinib (Standard) is the analytical standard of Cobimetinib. This product is intended for research and analytical applications. Cobimetinib (GDC-0973, RG7420) is a potent, selective and oral MEK1 inhibitor with an IC50 of 4.2 nM for MEK1.
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Cat. No.: HY-13078R
CAS No.: 934662-91-6
Synonyms: GDC-0973 racemate (Standard); XL518 racemate (Standard)
Target:  

MEK Reference Standards

Research Areas:  

Cancer

Cobimetinib (racemate) (Standard) is the analytical standard of Cobimetinib (racemate). This product is intended for research and analytical applications. Cobimetinib racemate (GDC-0973 racemate; XL518 racemate) is the racemate of Cobimetinib. Cobimetinib is a potent and selective MEK inhibitor.
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Cat. No.: HY-13079
CAS No.: 934660-94-3
Purity:  99.78%
Synonyms: GDC-0973 (R-enantiomer); XL-518 (R-enantiomer)
Target:  

MEK

Research Areas:  

Cancer

Cobimetinib R-enantiomer is the less active R-enantiomer of Cobimetinib. Cobimetinib is a potent and selective MEK inhibitor.
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Cat. No.: HY-13078S
Synonyms: GDC-0973-13C6 racemate; XL518-13C6 racemate
Cobimetinib- 13C6 (GDC-0973- 13C6; XL518- 13C6) racemate is the deuterium labeled Cobimetinib (racemate) (HY-13078) . Cobimetinib racemate (GDC-0973 racemate; XL518 racemate) is the racemate of Cobimetinib. Cobimetinib is a potent and selective MEK inhibitor .
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