3 Results for "

Linopirdine

" in MedChemExpress (MCE) Product Catalog:
Products (3)

3 Results for "Linopirdine" in MCE Product Catalog:

2
2 Cited Publications
Cat. No.: HY-W020468
CAS No.: 105431-72-9
Synonyms: DuP 996
Research Areas:  

Neurological Disease

Linopirdine (DuP 996) is an orally active, selective M-type K + current (IM; Kv7; KCNQ Channels) inhibitor with an IC50 of 2.4 μM. Linopirdine is a TRPV1 agonist. Linopirdine, a putative cognition enhancing agent, increases acetylcholine release in rat brain tissue .
loading...
    loading...
Cat. No.: HY-108576
CAS No.: 113168-57-3
Synonyms: DuP 996 dihydrochloride
Target:  

TRP Channel

Research Areas:  

Neurological Disease

Linopirdine dihydrochloride is a agonist of capsaicin receptor TRPV1. Linopirdine increases the intracellular calcium concentration in HEK293 cells. Linopirdine dihydrochloride exerts an excitatory action on mammalian nociceptors .
loading...
    loading...
Cat. No.: HY-W020468R
CAS No.: 105431-72-9
Synonyms: DuP 996 (Standard)
Linopirdine (DuP 996) is an orally active, selective M-type K+ current (IM; Kv7; KCNQ Channels) inhibitor with an IC50 of 2.4 μM. Linopirdine is a TRPV1 agonist. Linopirdine, a putative cognition enhancing agent, increases acetylcholine release in rat brain tissue .
loading...
    loading...