8 Results for "

Mosapride

" in MedChemExpress (MCE) Product Catalog:
Products (8)

8 Results for "Mosapride" in MCE Product Catalog:

6
6 Publications Verification
Cat. No.: HY-B0189
CAS No.: 112885-41-3
Synonyms: TAK-370; AS-4370
Mosapride is an orally active gastroenterokinetic compound. Mosapride is a 5HT4 agonist. Mosapride is a CYP inducer. Mosapride has a concentration-dependent inhibitory effect on Kv4.3, and its IC50 value is 15.2 μM. Mosapride can be used in the study of gastrointestinal diseases .
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6
6 Publications Verification
Cat. No.: HY-B0189A
CAS No.: 112885-42-4
Synonyms: TAK-370 citrate; AS-4370 citrate
Mosapride citrate is an orally active gastroenterokinetic compound. Mosapride citrate is a 5HT4 agonist. Mosapride citrate is a CYP inducer. Mosapride citrate has a concentration-dependent inhibitory effect on Kv4.3, and its IC50 value is 15.2 μM. Mosapride citrate can be used in the study of gastrointestinal diseases .
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6
6 Publications Verification
Cat. No.: HY-B0189B
CAS No.: 636582-62-2
Synonyms: TAK-370 citrate dihydrate; AS-4370 citrate dihydrate
Mosapride (TAK-370) citrate dehydrate is a gastroprokinetic agent with 5-hydroxytryptamine4 receptor agonist activity and has been widely used in the research of a variety of gastrointestinal disorders. Mosapride citrate dihydrate potently inhibits Kv4.3 in a concentration-dependent manner with IC50 values of 15.2 μM . Mosapride citrate dihydrateselectively stimulates upper GI motility in vivo .
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Cat. No.: HY-B0189AR
CAS No.: 112885-42-4
Synonyms: TAK-370 citrate (Standard); AS-4370 citrate (Standard)
Mosapride (citrate) (Standard) is the analytical standard of Mosapride (citrate). This product is intended for research and analytical applications. Mosapride citrate is an orally active gastroenterokinetic compound. Mosapride citrate is a 5HT4 agonist. Mosapride citrate is a CYP inducer. Mosapride citrate has a concentration-dependent inhibitory effect on Kv4.3, and its IC50 value is 15.2 μM. Mosapride citrate can be used in the study of gastrointestinal diseases .
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Cat. No.: HY-B0189S1
CAS No.: 1246820-66-5
Mosapride-d5 is the deuterium labeled Mosapride. Mosapride is a gastroprokinetic agent that acts as a selective 5HT4 agonist.
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Cat. No.: HY-148846
CAS No.: 1161443-73-7
Target:  

Drug Metabolite

Research Areas:  

Metabolic Disease

Mosapride N-Oxide is a major active metabolite of Mosapride. Mosapride is a gastroprokinetic agent that acts as a selective 5HT4 agonist.
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Cat. No.: HY-Z6430
CAS No.: 152013-26-8
Target:  

5-HT Receptor

Research Areas:  

Neurological Disease

Des-4-fluorobenzyl mosapride is the primary metabolite of Mosapride (HY-B0189). Mosapride is an orally active gastroenterokinetic compound and is a 5HT4 agonist.
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Cat. No.: HY-141757S
CAS No.: 1246814-79-8
Des-p-fluorobenzyl mosapride-d5 is the deuterium labeled Des-p-fluorobenzyl mosapride .
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