5 Results for "

Ritanserin

" in MedChemExpress (MCE) Product Catalog:
Products (5)

5 Results for "Ritanserin" in MCE Product Catalog:

3
3 Cited Publications
Cat. No.: HY-10791
CAS No.: 87051-43-2
Purity:  99.68%
Synonyms: R 55667
Ritanserin (R 55667) is a highly potent, relatively selective, orally active, long acting antagonist of 5-HT2 receptor, with an IC50 of 0.9 nM, less active on Histamine H1, Dopamine D2, Adrenergic α1, Adrenergic α2 receptors .
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Cat. No.: HY-101324A
CAS No.: 61655-58-1
Purity:  99.69%
Synonyms: CPP monohydrochloride
Target:  

5-HT Receptor

Research Areas:  

Neurological Disease

MK-212 monohydrochloride (CPP monohydrochloride) is an orally active, blood-brain barrier permeable agonist of 5-HT1C, 5-HT2 and 5-HT1A receptors. MK-212 monohydrochloride induces hyperthermia, nausea, arousal, irritability and restlessness, inhibits the elevation of plasma cortisol and prolactin, and reduces feelings of calmness and overall positive affect. MK-212 monohydrochloride mediates anxiety-like behaviors and motor inhibition. MK-212 monohydrochloride is applicable to research related to schizophrenia and anxiety disorders .
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Cat. No.: HY-148174
CAS No.: 93076-87-0
Target:  

DGK

Research Areas:  

Cancer

JNJ-3790339, a Ritanserin (HY-10791) analog, is a potent and selective diacylglycerol kinase (DGKα) inhibitor with an IC50 of 9.6 μM. JNJ-3790339 has induction of toxicity in malignant cells, and improves ability to upregulate T cell activation .
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Cat. No.: HY-10791R
CAS No.: 87051-43-2
Synonyms: R 55667 (Standard)
Ritanserin (Standard) is the analytical standard of Ritanserin. This product is intended for research and analytical applications. Ritanserin (R 55667) is a highly potent, relatively selective, orally active, long acting antagonist of 5-HT2 receptor, with an IC50 of 0.9 nM, less active on Histamine H1, Dopamine D2, Adrenergic α1, Adrenergic α2 receptors .
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Cat. No.: HY-101324
CAS No.: 64022-27-1
Synonyms: CPP
Target:  

5-HT Receptor

Research Areas:  

Neurological Disease

MK-212 (CPP) is an orally active, blood-brain barrier permeable agonist of 5-HT1C, 5-HT2 and 5-HT1A receptors. MK-212 induces hyperthermia, nausea, arousal, irritability and restlessness, inhibits the elevation of plasma cortisol and prolactin, and reduces feelings of calmness and overall positive affect. MK-212 mediates anxiety-like behaviors and motor inhibition. MK-212 is applicable to research related to schizophrenia and anxiety disorders .
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