9 Results for "

Rizatriptan

" in MedChemExpress (MCE) Product Catalog:
Products (9)

9 Results for "Rizatriptan" in MCE Product Catalog:

Cat. No.: HY-B0206
CAS No.: 145202-66-0
Synonyms: MK 462
Target:  

5-HT Receptor

Research Areas:  

Neurological Disease

Rizatriptan benzoate is the agonist for 5-HT1B and 5-HT1D. Rizatriptan benzoate has a peripheral vasoconstrictive effect, penetrates the intact blood-brain barrier, and inhibits pain neurotransmission in the central nervous system .
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Cat. No.: HY-B0206R
CAS No.: 145202-66-0
Synonyms: MK 462 (Standard)
Research Areas:  

Neurological Disease

Rizatriptan (benzoate) (Standard) is the analytical standard of Rizatriptan (benzoate). This product is intended for research and analytical applications. Rizatriptan benzoate is the agonist for 5-HT1B and 5-HT1D. Rizatriptan benzoate has a peripheral vasoconstrictive effect, penetrates the intact blood-brain barrier, and inhibits pain neurotransmission in the central nervous system .
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Cat. No.: HY-W018475
CAS No.: 144034-80-0
Synonyms: MK 462 free base
Target:  

5-HT Receptor

Research Areas:  

Neurological Disease

Rizatriptan (MK 462 free base) is an orally active 5-HT1B/5-HT1D receptor agonist, with BBB permeability. Rizatriptan exerts significant anti-migraine effects by constricting intracranial and extracranial blood vessels and inhibiting neuropeptide release. Rizatriptan exhibits species- and tissue-specific metabolic characteristics; for example, it undergoes oxidative deamination mainly by MAO-A in the liver of brown rats, so co-administration with MAO-A inhibitors is prohibited. Rizatriptan may also exacerbate nitroglycerin-induced cutaneous allodynia, prolong the duration of central sensitization, and increase anxiety-like behavior and active drug-seeking behavior in mice. Rizatriptan has been widely used in studies related to migraine and medication-overuse headache .
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Cat. No.: HY-Z8410
CAS No.: 260435-42-5
Target:  

Drug Derivative

Research Areas:  

Others

Rizatriptan N-oxide is the impurity of Rizatriptan.
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Cat. No.: HY-B0206S
CAS No.: 1216984-85-8
Rizatriptan-d6 (benzoate) is the deuterium labeled Rizatriptan benzoate. Rizatriptan benzoate is the agonist for 5-HT1B and 5-HT1D. Rizatriptan benzoate has a peripheral vasoconstrictive effect, penetrates the intact blood-brain barrier, and inhibits pain neurotransmission in the central nervous system .
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Cat. No.: HY-W018475B
CAS No.: 159776-67-7
Synonyms: MK 462 hemisulfate hemihydrate
Target:  

5-HT Receptor

Research Areas:  

Neurological Disease

Rizatriptan (MK 462) hemisulfate hemihydrate is the agonist for 5-HT1B and 5-HT1D. Rizatriptan hemisulfate hemihydrate has a peripheral vasoconstrictive effect, penetrates the intact blood-brain barrier, and inhibits pain neurotransmission in the central nervous system .
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Cat. No.: HY-W700240
CAS No.: 177270-91-6
Target:  

5-HT Receptor

Research Areas:  

Neurological Disease

Triazolomethylindole-3-acetic acid is a metabolite of the serotonin (5-HT) receptor subtype 5-HT1B and 5-HT1D agonist Rizatriptan HY-B0206).
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Cat. No.: HY-132432S
CAS No.: 1215678-02-6
N10-Monodesmethyl Rizatriptan-d3 is the deuterium labeled N10-Monodesmethyl Rizatriptan .
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Cat. No.: HY-132440S
CAS No.: 1329834-30-1
Synonyms: N,N-Dimethyl-5-(1H-1,2,4-triazol-1-ylmethyl)-1H-indole-2-ethanamine-d6
Iso Rizatriptan-d6 is the deuterium labeled Iso Rizatriptan .
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