5 Results for "

Sabcomeline

" in MedChemExpress (MCE) Product Catalog:
Products (5)

5 Results for "Sabcomeline" in MCE Product Catalog:

Cat. No.: HY-106432A
CAS No.: 159912-58-0
Purity:  99.86%
Synonyms: SB-202026 hydrochloride; Memric hydrochloride
Target:  

mAChR Dopamine Receptor

Research Areas:  

Neurological Disease

Sabcomeline (SB-202026; Memric) hydrochloride is a muscarinic receptor agonist capable of crossing the blood-brain barrier. Sabcomeline hydrochloride exhibits affinity for all hM1 to hM5 subtypes (pKi=6.72-7.23), and shows near-full agonism at the hM3 receptor, inducing extracellular acidification. Sabcomeline hydrochloride alters the binding kinetics of dopamine D2 receptors through neural network regulation. Sabcomeline hydrochloride also causes minimal cardiovascular changes, effectively reverses spatial memory deficits in rodents and induces conditioned taste aversion. Sabcomeline hydrochloride is an important tool compound in studies of Alzheimer's disease and related neurodegenerative diseases .
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Cat. No.: HY-106432
CAS No.: 159912-53-5
Synonyms: SB-202026; Memric
Target:  

mAChR

Research Areas:  

Neurological Disease

Sabcomeline (SB-202026) is a potent and functionally selective muscarinic M1 receptor partial agonist that improve cognition. Sabcomeline can be used for Alzheimer's disease research .
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Cat. No.: HY-167933
CAS No.: 133642-67-8
Synonyms: (Rac)-SB-202026 hydrochloride; (Rac)-Memric hydrochloride
Target:  

mAChR

Research Areas:  

Neurological Disease

(Rac)-Sabcomeline ((Rac)-SB-202026) hydrochloride serves as an M1 receptor agonist, making it a valuable tool for research into Alzheimer's disease.
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Cat. No.: HY-167947
CAS No.: 149156-36-5
Synonyms: (Rac)-SB-202026; (Rac)-Memric
Target:  

mAChR

Research Areas:  

Neurological Disease

(Rac)-Sabcomeline ((Rac)-SB-202026) serves as an M1/M4 muscarinic agonist, making it a valuable tool in the exploration of neurological disorders, including schizophrenia.
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Cat. No.: HY-106432AR
CAS No.: 159912-58-0
Synonyms: SB-202026 hydrochloride (Standard); Memric hydrochloride (Standard)
Research Areas:  

Neurological Disease

Sabcomeline hydrochloride (Standard) is the analytical standard of Sabcomeline hydrochloride (HY-106432A). This product is intended for research and analytical applications. Sabcomeline (SB-202026) hydrochloride is a potent and functionally selective muscarinic M1 receptor partial agonist that improve cognition. Sabcomeline hydrochloride can be used for Alzheimer's disease research .
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