SSTR4 agonist 5
SSTR4 agonist 5 (Compound 5) is the orally active agonist for somatostatin receptor 4 (SSTR4) with an EC50 of 0.228 nM. SSTR4 agonist 5 exhibits good stability in human/rat liver microsomes. SSTR4 agonist 5 inhibits mechanical hyperalgesia in rat models.
For research use only. We do not sell to patients.
- CAS No.: 2761347-44-6
- Formula: C20H26N4O
- Molecular Weight:338.45
-
Storage:
Please store the product under the recommended conditions in the Certificate of Analysis.
Biological Activity
|
SSTR4 0.228 nM (IC50) |
Chemical Information
-
CAS No. 2761347-44-6
-
Molecular Weight 338.45
-
Formula C20H26N4O
-
SMILES
O=C(C1C2CNCC12C)NC(C)(C)C3=NC4=C5C(CCC4)=CC=CN35
-
Shipping
Room temperature in continental US; may vary elsewhere.
-
Storage
Please store the product under the recommended conditions in the Certificate of Analysis.
Purity & Documentation
References
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)