SSTR5 antagonist 3
SSTR5 antagonist 3 (Compound 23) is an orally active somatostatin receptor subtype 5 (SSTR5) antagonist with low hERG inhibition. SSTR5 antagonist 3 exhibits potency with IC50 values of 2.8 nM and 1.4 nM in human and mouse, respectively. SSTR5 antagonist 3 can be used for the research of anti-gallstone.
For research use only. We do not sell to patients.
- CAS No.: 2851454-42-5
- Formula: C31H36F2N2O5
- Molecular Weight:554.62
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Storage:
Please store the product under the recommended conditions in the Certificate of Analysis.
Biological Activity
IC50: 2.8 nM (human); 1.4 nM (mouse)[1].
Chemical Information
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CAS No. 2851454-42-5
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Molecular Weight 554.62
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Formula C31H36F2N2O5
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SMILES
FC1=CC=C(C2=C(C=C(C=C2OCC)CN3CCC(F)(CC3)CNC4=CC(OC)=C(C(O)=O)C=C4)OCC)C=C1
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Shipping
Room temperature in continental US; may vary elsewhere.
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Storage
Please store the product under the recommended conditions in the Certificate of Analysis.
Purity & Documentation
References
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)