1. GPCR/G Protein
  2. Angiotensin Receptor
  3. Azilsartan-d5

Azilsartan-d5  (Synonyms: TAK-536-d5)

Cat. No.: HY-14914S Purity: 99.42%
COA Handling Instructions

Azilsartan-d5 is the deuterium labeled Azilsartan(TAK-536), which is a specific and potent angiotensin II type 1 receptor antagonist.

For research use only. We do not sell to patients.

Azilsartan-d<sub>5</sub> Chemical Structure

Azilsartan-d5 Chemical Structure

CAS No. : 1346599-45-8

Size Price Stock Quantity
Solid + Solvent
10 mM * 1 mL in DMSO
ready for reconstitution
USD 832 In-stock
Solution
10 mM * 1 mL in DMSO USD 832 In-stock
Solid
1 mg USD 195 In-stock
5 mg USD 820 In-stock
10 mg   Get quote  
50 mg   Get quote  

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Based on 1 publication(s) in Google Scholar

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Description

Azilsartan-d5 is the deuterium labeled Azilsartan(TAK-536), which is a specific and potent angiotensin II type 1 receptor antagonist.

Molecular Weight

461.48

Formula

C25H15D5N4O5

CAS No.
Appearance

Solid

Color

White to off-white

SMILES

OC(C1=CC=CC2=C1N(C(OC(C([2H])([2H])[2H])([2H])[2H])=N2)CC(C=C3)=CC=C3C4=CC=CC=C4C5=NC(ON5)=O)=O

Shipping

Room temperature in continental US; may vary elsewhere.

Storage
Powder -20°C 3 years
4°C 2 years
In solvent -80°C 2 years
-20°C 1 year
Solvent & Solubility
In Vitro: 

DMSO : 100 mg/mL (216.69 mM; Need ultrasonic; Hygroscopic DMSO has a significant impact on the solubility of product, please use newly opened DMSO)

Preparing
Stock Solutions
Concentration Solvent Mass 1 mg 5 mg 10 mg
1 mM 2.1669 mL 10.8347 mL 21.6694 mL
5 mM 0.4334 mL 2.1669 mL 4.3339 mL
View the Complete Stock Solution Preparation Table

* Please refer to the solubility information to select the appropriate solvent. Once prepared, please aliquot and store the solution to prevent product inactivation from repeated freeze-thaw cycles.
Storage method and period of stock solution: -80°C, 2 years; -20°C, 1 year. When stored at -80°C, please use it within 2 years. When stored at -20°C, please use it within 1 year.

  • Molarity Calculator

  • Dilution Calculator

Mass (g) = Concentration (mol/L) × Volume (L) × Molecular Weight (g/mol)

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Molecular Weight *

Concentration (start) × Volume (start) = Concentration (final) × Volume (final)

This equation is commonly abbreviated as: C1V1 = C2V2

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Volume (start)

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C2

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V2

In Vivo Dissolution Calculator
Please enter the basic information of animal experiments:

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Recommended: Prepare an additional quantity of animals to account for potential losses during experiments.
Calculation results:
Working solution concentration: mg/mL
Purity & Documentation

Purity: 99.42%

References

Complete Stock Solution Preparation Table

* Please refer to the solubility information to select the appropriate solvent. Once prepared, please aliquot and store the solution to prevent product inactivation from repeated freeze-thaw cycles.
Storage method and period of stock solution: -80°C, 2 years; -20°C, 1 year. When stored at -80°C, please use it within 2 years. When stored at -20°C, please use it within 1 year.

Optional Solvent Concentration Solvent Mass 1 mg 5 mg 10 mg 25 mg
DMSO 1 mM 2.1669 mL 10.8347 mL 21.6694 mL 54.1735 mL
5 mM 0.4334 mL 2.1669 mL 4.3339 mL 10.8347 mL
10 mM 0.2167 mL 1.0835 mL 2.1669 mL 5.4174 mL
15 mM 0.1445 mL 0.7223 mL 1.4446 mL 3.6116 mL
20 mM 0.1083 mL 0.5417 mL 1.0835 mL 2.7087 mL
25 mM 0.0867 mL 0.4334 mL 0.8668 mL 2.1669 mL
30 mM 0.0722 mL 0.3612 mL 0.7223 mL 1.8058 mL
40 mM 0.0542 mL 0.2709 mL 0.5417 mL 1.3543 mL
50 mM 0.0433 mL 0.2167 mL 0.4334 mL 1.0835 mL
60 mM 0.0361 mL 0.1806 mL 0.3612 mL 0.9029 mL
80 mM 0.0271 mL 0.1354 mL 0.2709 mL 0.6772 mL
100 mM 0.0217 mL 0.1083 mL 0.2167 mL 0.5417 mL
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Azilsartan-d5 Related Classifications

Help & FAQs
  • Do most proteins show cross-species activity?

    Species cross-reactivity must be investigated individually for each product. Many human cytokines will produce a nice response in mouse cell lines, and many mouse proteins will show activity on human cells. Other proteins may have a lower specific activity when used in the opposite species.

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