2. GPCR/G Protein
  3. RXFP Receptor
  4. RXFP3/4 agonist 1

RXFP3/4 agonist 1 is an agonist of relaxin family peptide 3/4 receptor (RXFP3/4), with EC50s of 82/2 nM, respectivley. RXFP3/4 agonist 1 increases food intake in rats.

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RXFP3/4 agonist 1 Chemical Structure

RXFP3/4 agonist 1 Chemical Structure

CAS No. : 2351104-40-8

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RXFP3/4 agonist 1 Related Antibodies

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Description

RXFP3/4 agonist 1 is an agonist of relaxin family peptide 3/4 receptor (RXFP3/4), with EC50s of 82/2 nM, respectivley. RXFP3/4 agonist 1 increases food intake in rats[1].

IC50 & Target

EC50: 82 nM (RXFP3), 2 nM (RXFP4)[1]
In Vitro

RXFP3/4 agonist 1 (Compound 4) inhibits orskolin-stimulated cAMP accumulation in CHO-K1 cells stably overexpressing RXFP3 and RXFP4, with EC50s of 12.8 and 1.6 nM, respectively[1].

MedChemExpress (MCE) has not independently confirmed the accuracy of these methods. They are for reference only.

RXFP3/4 agonist 1 Related Antibodies
Molecular Weight

383.87

Formula

C20H22ClN5O
CAS No.
SMILES

CCC1=C(NC=C2/C=N/NC(NCCC3=CC=C(Cl)C=C3)=N)C2=CC(O)=C1
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Room temperature in continental US; may vary elsewhere.
Storage

Please store the product under the recommended conditions in the Certificate of Analysis.
Purity & Documentation
References
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RXFP3/4 agonist 1 Related Classifications

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Help & FAQs
  • Do most proteins show cross-species activity?

    Species cross-reactivity must be investigated individually for each product. Many human cytokines will produce a nice response in mouse cell lines, and many mouse proteins will show activity on human cells. Other proteins may have a lower specific activity when used in the opposite species.

Keywords:

RXFP3/4 agonist 12351104-40-8RXFP ReceptorInhibitorinhibitorinhibit

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RXFP3/4 agonist 1
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