1. Signaling Pathways
  2. GPCR/G Protein
  3. Bradykinin Receptor
  4. Bradykinin B2 Receptor (B2R) Isoform
  5. Bradykinin B2 Receptor (B2R) Antagonist

Bradykinin B2 Receptor (B2R) Antagonist

Bradykinin B2 Receptor (B2R) Antagonists (4):

Cat. No. Product Name Effect Purity
  • HY-17446
    Icatibant
    Antagonist 99.51%
    Icatibant (HOE-140) is a potent and specific peptide antagonist of bradykinin B2 receptor with IC50 and Ki of 1.07 nM and 0.798 nM respectively.
  • HY-106277
    Fasitibant free base
    Antagonist
    Fasitibant (free base) is a potent, selective, high affinity, and long-lasting nonpeptide bradykinin B2 (BK2) receptor antagonist. Fasitibant (free base) has proinflammatory effects and can be used for the research of osteoarthritis and rheumatoid arthritis.
  • HY-P3232
    B 9430
    Antagonist
    B 9430 is a potent bradykinin B1/B2 receptor antagonist.
  • HY-106277A
    Fasitibant chloride hydrochloride
    Antagonist
    Fasitibant chloride hydrochloride (MEN16132) is a potent, selective, high affinity, and long-lasting nonpeptide bradykinin B2 (BK2) receptor antagonist. Fasitibant chloride hydrochloride has proinflammatory effects and can be used for the research of osteoarthritis and rheumatoid arthritis.