Drug Derivative
Drug derivative
Drug derivatives are derived from parent compounds. They replace or add atoms and groups through chemical reactions to optimize the various properties of the parent compound and reduce side effects. The application of drug derivatives provides a diverse compound library for drug research and development and accelerates the discovery of new drugs. For example, urea derivatives Glibenclamide can prolong the blood sugar-lowering effect of anti-diabetic drugs.
References:
- [1]. Vardanyan RS, et al. Fentanyl-related compounds and derivatives: current status and future prospects for pharmaceutical applications. Future Med Chem. 2014 Mar;6(4):385-412.x
- [2]. Ghosh AK, et al. Urea Derivatives in Modern Drug Discovery and Medicinal Chemistry. J Med Chem. 2020 Mar 26;63(6):2751-2788.x
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Drug Derivative Related Products (4062)
Related Products (4062)
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Ingenol 3-Hexanoate
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K-TMZ
0 ImagesCat. No.: HY-115690CAS No.: 2269482-26-8K-TMZ is a derivative of methyl ketone, which exhibits antitumor efficacy against O6 -methylguanine DNA methyltransferase (MGMT) deficient cell. K-TMZ can be used for research of glioblastoma.
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1-Propinoyl Lysergic acid methylisopropylamide
0 ImagesCat. No.: HY-150342CAS No.: 3028950-73-1Synonyms: 1P-MiPLA1-Propinoyl Lysergic acid methylisopropylamide (1P-MiPLA) is a lysergamide compound.
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Dimethyl octadecanedioate
0 ImagesSynonyms: Octadecanedioic acid,dimethyl esterDimethyl octadecanedioate (Octadecanedioic acid,dimethyl ester) is an ester product.
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L-Ascorbyl myristate
0 ImagesCat. No.: HY-121860CAS No.: 33425-76-2L-Ascorbyl myristate is a bioactive compound with notable chemical properties.
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D-19050
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WAY-649123
0 ImagesWAY-649123 is an active molecule.
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3',4'-Trimethylene-α-methylamino-valerophenone hydrochloride
0 ImagesCat. No.: HY-175126CAS No.: 2749282-62-83',4'-Trimethylene-α-methylamino-valerophenone hydrochloride is a drug analogue, which can be used in the research of neurological diseases.
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LY-295501
0 ImagesCat. No.: HY-169129CAS No.: 150869-74-2Synonyms: ILX-295501
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WAY-313318
0 ImagesWAY-313318 is an active molecule.
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Methyl heptadecanoate (Standard)
0 ImagesCat. No.: HY-W004290RCAS No.: 1731-92-6Synonyms: Methyl margarate (Standard)Methyl heptadecanoate (Standard) is the analytical standard of Methyl heptadecanoate (HY-W004290). This product is intended for research and analytical applications. Methyl heptadecanoate (C17:0 methyl ester) is the methyl ester derivative of heptadecanoic acid (HY-W004284). Methyl heptadecanoate is used as an internal standard for quantitative calibration of fatty acids in GC-MS analysis.
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4-Benzylphenol
0 ImagesCat. No.: HY-W091820CAS No.: 101-53-1Synonyms: 4HDPM4-Benzylphenol (4HDPM), a structural analog of Bisphenol F (HY-W014901), has estrogenic activity in vitro and in vivo. 4-Benzylphenol can be used in plastics as a germicide, antiseptic, preservative, and antioxidant, and can be used in during organic synthesis.
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rel-FTY720 phenoxy-biotin hydrochloride
0 ImagesCat. No.: HY-181455CAS No.: 2309930-88-7rel-FTY720 phenoxy-biotin hydrochloride is a chemical probe designed based on the structure of Fingolimod (HY-12005), which incorporates a phenoxy group capable of specific click chemistry reactions and is conjugated with a biotin tag.
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Mesuagin
0 ImagesCat. No.: HY-N9650CAS No.: 21721-08-4Synonyms: Mammea A/AD cyclo DMesuagin (Mammea A/AD cyclo D) shows anticancer activity and can be isolated from the Mammea americana L. seeds.
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N-Butyl Pentedrone hydrochloride
0 ImagesCat. No.: HY-150340CAS No.: 18268-13-8N-Butyl Pentedrone hydrochloride is a drug derivative.
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N-Ethyl-4-methoxyamphetamine hydrochloride
0 ImagesCat. No.: HY-W280622CAS No.: 93963-24-7N-Ethyl-4-methoxyamphetamine hydrochloride is an analog of 4-Methoxyamphetamine. The addition of an N-ethyl substituent decreases analgesic potency.
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2-BZP
0 ImagesCat. No.: HY-60174CAS No.: 84477-71-4Synonyms: 2-Benzylpiperazin2-BZP is a piperazine.
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Antitumor agent-160
0 ImagesCat. No.: HY-W781271CAS No.: 1262489-36-0Antitumor agent-160 (compound Ia) is a derivative of the antifungal agent PHENALENONE (HY-W286805) and has antitumor activity.
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Tetrahydrocannabivarin acetate
0 ImagesCat. No.: HY-168362CAS No.: 885123-57-9Synonyms: 1-Acetyl-△9-THCVTetrahydrocannabivarin acetate (1-Acetyl-△9-THCV) is structurally similar to known phytocannabinoids.
